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b synthesis

5synthesis methods
-

Yield:752242-26-5 99%

Reaction Conditions:

with potassium carbonate in N,N-dimethyl-formamide at 60;

References:

Iino, Tomoharu;Tsukahara, Daisuke;Kamata, Kenji;Sasaki, Kaori;Ohyama, Sumika;Hosaka, Hideka;Hasegawa, Takuro;Chiba, Masato;Nagata, Yasufumi;Eiki, Jun-ichi;Nishimura, Teruyuki [Bioorganic and Medicinal Chemistry,2009,vol. 17,# 7,p. 2733 - 2743] Location in patent:experimental part