(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE

132861-87-1

CAS-Nr.: 132861-87-1

Englisch Name:: (2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE

Synonyma:: PD 81,723;4,5-Dimethyl-3-[3-(trifluoromethyl)benzoyl]-2-thiophenamine;(2-Amino-4,5-dimethylthiophen-3-yl)(3-trifluoromethylphenyl) ketone;(3-Trifluoromethylphenyl)(2-amino-4-methyl-5-methyl-3-thienyl) ketone;(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE;Methanone, (2-aMino-4,5-diMethyl-3-thienyl)[3-(trifluoroMethyl)phenyl]-;(2-amino-4,5-dimethyl-3-thiophenyl)-[3-(trifluoromethyl)phenyl]methanone;(2-Amino-4,5-dimethylthiophen-3-yl)-(3-(trifluoromethyl)phenyl)methanone

CBNumber:: CB2484082

Summenformel:: C14H12F3NOS

Molgewicht:: 299.31

MOL-Datei:: 132861-87-1.mol

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Eigenschaften Sicherheit Verwendungswort Produktionsfirma 38

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Eigenschaften

Schmelzpunkt:: 100-104 °C(Solv: ligroine (8032-32-4))

Siedepunkt:: 411.7±45.0 °C(Predicted)

Dichte: 1.328±0.06 g/cm3(Predicted)

storage temp.: Sealed in dry,2-8°C

Löslichkeit: DMSO: ~13 mg/mL

Aggregatzustand: solid

pka: -1.36±0.13(Predicted)

Farbe: yellow

Sicherheit

WGK Germany	3

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Chemische Eigenschaften,Einsatz,Produktion Methoden

Verwenden

PD 81,723 is an allosteric potentiator that increases the functional effects of adenosine and adenosine analogs.

Biologische Aktivität

Allosteric potentiator at the adenosine A 1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t 1/2 of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A 1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo .

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Upstream-Materialien And Downstream Produkte

Upstream-Materialien

Downstream Produkte

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Anbieter Lieferant Produzent Hersteller Vertrieb Händler.

Global( 38)Lieferanten

Firmenname	Telefon	E-Mail	Land	Produktkatalog	Edge Rate
Alchem Pharmtech,Inc.	8485655694	sales@alchempharmtech.com	United States	63711	58
TargetMol Chemicals Inc.	+1-781-999-5354 +1-00000000000	marketing@targetmol.com	United States	19892	58
Aladdin Scientific	+1-+1(833)-552-7181	sales@aladdinsci.com	United States	52927	58
Amadis Chemical Company Limited	571-89925085	sales@amadischem.com	China	131980	58
3B Pharmachem (Wuhan) International Co.,Ltd.	821-50328103-801 18930552037	3bsc@sina.com	China	15848	69
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8449	60
Aikon International Limited	025-58859352 18068836627	sales01@aikonchem.com	China	15085	58
BOC Sciences	--	info@bocsci.com	USA	0	65
Energy Chemical	021-58432009 400-005-6266	marketing1@energy-chemical.com	China	44844	58
Shanghai Universal Biotech Co.,Ltd	13774214275	gaojun@univ-bio.com	China	24990	58

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE
PD 81,723
(2-Amino-4,5-dimethylthiophen-3-yl)(3-trifluoromethylphenyl) ketone
(3-Trifluoromethylphenyl)(2-amino-4-methyl-5-methyl-3-thienyl) ketone
4,5-Dimethyl-3-[3-(trifluoromethyl)benzoyl]-2-thiophenamine
Methanone, (2-aMino-4,5-diMethyl-3-thienyl)[3-(trifluoroMethyl)phenyl]-
(2-Amino-4,5-dimethylthiophen-3-yl)-(3-(trifluoromethyl)phenyl)methanone
(2-amino-4,5-dimethyl-3-thiophenyl)-[3-(trifluoromethyl)phenyl]methanone
132861-87-1
C14H12F3NOS
Adenosine receptor