(2-아미노-4,5-디메틸-3-티에닐)-[3-(트리플루오로메틸)페닐]메타논 C화학적 특성, 용도, 생산
용도
PD 81,723 is an allosteric potentiator that increases the functional effects of adenosine and adenosine analogs.
생물학적 활성
Allosteric potentiator at the adenosine A 1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t 1/2 of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A 1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo .
(2-아미노-4,5-디메틸-3-티에닐)-[3-(트리플루오로메틸)페닐]메타논 준비 용품 및 원자재