ChemicalBook >> CAS DataBase List >>(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE

CAS No.
132861-87-1
Chemical Name:
(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE
Synonyms
PD 81,723;4,5-Dimethyl-3-[3-(trifluoromethyl)benzoyl]-2-thiophenamine;(2-Amino-4,5-dimethylthiophen-3-yl)(3-trifluoromethylphenyl) ketone;(3-Trifluoromethylphenyl)(2-amino-4-methyl-5-methyl-3-thienyl) ketone;(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE;Methanone, (2-aMino-4,5-diMethyl-3-thienyl)[3-(trifluoroMethyl)phenyl]-;(2-amino-4,5-dimethyl-3-thiophenyl)-[3-(trifluoromethyl)phenyl]methanone;(2-Amino-4,5-dimethylthiophen-3-yl)-(3-(trifluoromethyl)phenyl)methanone
CBNumber:
CB2484082
Molecular Formula:
C14H12F3NOS
Molecular Weight:
299.31
MDL Number:
MFCD01321053
MOL File:
132861-87-1.mol
Last updated:2024-10-23 13:36:13

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Properties

Melting point 100-104 °C(Solv: ligroine (8032-32-4))
Boiling point 411.7±45.0 °C(Predicted)
Density 1.328±0.06 g/cm3(Predicted)
storage temp. Sealed in dry,2-8°C
solubility DMSO: ~13 mg/mL
form solid
pka -1.36±0.13(Predicted)
color yellow

SAFETY

Risk and Safety Statements

WGK Germany  3

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE price More Price(16)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Tocris 1363 PD 81,723 ≥99%(HPLC) 132861-87-1 10 $157 2021-12-16 Buy
Usbiological 256193 PD 81723 132861-87-1 10mg $403 2021-12-16 Buy
TRC P218318 PD 81,723 132861-87-1 10mg $115 2021-12-16 Buy
Matrix Scientific 096431 (2-Amino-4,5-dimethylthiophen-3-yl)-(3-(trifluoromethyl)phenyl)methanone 95+% 132861-87-1 250mg $1890 2021-12-16 Buy
AK Scientific 6013AA (2-Amino-4,5-dimethylthiophen-3-yl)(3-(trifluoromethyl)phenyl)methanone 132861-87-1 250mg $2601 2021-12-16 Buy
Product number Packaging Price Buy
1363 10 $157 Buy
256193 10mg $403 Buy
P218318 10mg $115 Buy
096431 250mg $1890 Buy
6013AA 250mg $2601 Buy

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Chemical Properties,Uses,Production

Uses

PD 81,723 is an allosteric potentiator that increases the functional effects of adenosine and adenosine analogs.

Biological Activity

Allosteric potentiator at the adenosine A 1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t 1/2 of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A 1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo .

storage

Store at RT

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Preparation Products And Raw materials

Raw materials

Preparation Products

(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE Suppliers

Global( 38)Suppliers
Supplier Tel Email Country ProdList Advantage
Alchem Pharmtech,Inc.
8485655694 sales@alchempharmtech.com United States 63687 58
TargetMol Chemicals Inc.
+1-781-999-5354 +1-00000000000 marketing@targetmol.com United States 32165 58
Aladdin Scientific
+1-+1(833)-552-7181 sales@aladdinsci.com United States 52925 58
Amadis Chemical Company Limited
571-89925085 sales@amadischem.com China 131957 58
3B Pharmachem (Wuhan) International Co.,Ltd. 821-50328103-801 18930552037 3bsc@sina.com China 15839 69
EMMX Biotechnology LLC 888-539-0666 info@emmx.com United States 8447 60
Aikon International Limited 025-58859352 18068836627 sales01@aikonchem.com China 15084 58
BOC Sciences -- info@bocsci.com USA 0 65
Energy Chemical 021-58432009 400-005-6266 marketing1@energy-chemical.com China 44808 58
Shanghai Universal Biotech Co.,Ltd 13774214275 zhouzz@univ-bio.com China 24990 58

View Lastest Price from (2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
PD 81723 pictures 2024-10-24 PD 81723
132861-87-1
US $1970.00-488.00 / mg 10g TargetMol Chemicals Inc.
  • PD 81723 pictures
  • PD 81723
    132861-87-1
  • US $1970.00-488.00 / mg
  • TargetMol Chemicals Inc.
(2-AMINO-4,5-DIMETHYL-3-THIENYL)-[3-(TRIFLUOROMETHYL)PHENYL]METHANONE PD 81,723 (2-Amino-4,5-dimethylthiophen-3-yl)(3-trifluoromethylphenyl) ketone (3-Trifluoromethylphenyl)(2-amino-4-methyl-5-methyl-3-thienyl) ketone 4,5-Dimethyl-3-[3-(trifluoromethyl)benzoyl]-2-thiophenamine Methanone, (2-aMino-4,5-diMethyl-3-thienyl)[3-(trifluoroMethyl)phenyl]- (2-Amino-4,5-dimethylthiophen-3-yl)-(3-(trifluoromethyl)phenyl)methanone (2-amino-4,5-dimethyl-3-thiophenyl)-[3-(trifluoromethyl)phenyl]methanone 132861-87-1 C14H12F3NOS Adenosine receptor