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PD 135158

PD 135158 Structure
CAS No.
130325-35-8
Chemical Name:
PD 135158
Synonyms
PD 135158;4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid
CBNumber:
CB41400397
Molecular Formula:
C42H61N5O11
Molecular Weight:
811.97
MOL File:
130325-35-8.mol
Modify Date:
2023/5/18 11:31:03
Request For Quotation

PD 135158 Properties

storage temp. Store at +4°C
solubility <61.68mg/ml in DMSO

PD 135158 Chemical Properties,Uses,Production

Biological Activity

Potent and selective, nonpeptide CCK 2 receptor antagonist (IC 50 values are 2.8 and 1232 nM for CCK 2 and CCK 1 respectively) that displays negligible affinity at GABA A , benzodiazepine, substance P, neurotensin, opioid, bradykinin and 5-HT 3 receptors (IC 50 > 10 μ M). Exhibits anxiolytic activity in elevated plus maze and social interaction tests and increases food intake in rats.

PD 135158 Preparation Products And Raw materials

Raw materials

Preparation Products

PD 135158 Suppliers

Global( 16)Suppliers
Supplier Tel Country ProdList Advantage Inquiry
TargetMol Chemicals Inc. +1-781-999-5354 +1-00000000000 United States 19892 58 Inquiry
Tocris Bioscience +44 (0) 117 916 3333 United Kingdom 5729 77 Inquiry
3B Pharmachem (Wuhan) International Co.,Ltd. 821-50328103-801 18930552037 China 15848 69 Inquiry
ApexBio Technology + 1-832-696-8203 United States 6254 58 Inquiry
Beijing Baiao Innovation Technology Co., Ltd. 010-5718533 13366620421 CHINA 6005 58 Inquiry
Qingdao Jieshikang Biotechnology Co., Ltd. 4009025885 18754289606 CHINA 4012 58 Inquiry
Shanghai Haoyang Biological Technology Co., Ltd. 021-54046790 15121098156 CHINA 2905 58 Inquiry
Shanghai Weiwei Biological Technology Co., Ltd. 021-55669583 18616258598 CHINA 4398 58 Inquiry
Shanghai Chaoyan Biotechnology Co., Ltd. 021-50840550 CHINA 6217 58 Inquiry
Shanghai Hao Biological Technology Co., Ltd. 021-80370006 13585899102 CHINA 6805 58 Inquiry
Supplier Advantage
TargetMol Chemicals Inc. 58
Tocris Bioscience 77
3B Pharmachem (Wuhan) International Co.,Ltd. 69
ApexBio Technology 58
Beijing Baiao Innovation Technology Co., Ltd. 58
Qingdao Jieshikang Biotechnology Co., Ltd. 58
Shanghai Haoyang Biological Technology Co., Ltd. 58
Shanghai Weiwei Biological Technology Co., Ltd. 58
Shanghai Chaoyan Biotechnology Co., Ltd. 58
Shanghai Hao Biological Technology Co., Ltd. 58

130325-35-8(PD 135158)Related Search:

PD 135158 endo-1,7,7-Trimethylbicyclo(2.2.1)-2-heptanol, 97% L(-)-Borneol BORNYL FORMATE
PD 135158 4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid 130325-35-8