THIOPERAMIDE MALEATE
![THIOPERAMIDE MALEATE Structure](CAS/GIF/106243-16-7.gif)
- CAS No.
- 106243-16-7
- Chemical Name:
- THIOPERAMIDE MALEATE
- Synonyms
- Thiop;MR 12842;thioperamide;THIOPERAMIDE MALEATE;THIOPERAMIDE MALEATE SALT;THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE;N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide;N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide;N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE;N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
- CBNumber:
- CB5245732
- Molecular Formula:
- C15H24N4S
- Molecular Weight:
- 292.44
- MOL File:
- 106243-16-7.mol
- MSDS File:
- SDS
- Modify Date:
- 2023/6/30 15:45:59
THIOPERAMIDE MALEATE Chemical Properties,Uses,Production
Uses
Thioperamide is a highly potent and selective ligand for histamine H3-receptors.
Biological Activity
Potent histamine H 3 and H 4 antagonist/inverse agonist. K i values are 25 and 27 nM for human recombinant H 3 and H 4 receptors respectively. Blocks eosinophil shape change (IC 50 = 1.4 μ M) and chemotaxis (IC 50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H 3 Receptor Tocriset™ .
THIOPERAMIDE MALEATE Preparation Products And Raw materials
Raw materials
Preparation Products
THIOPERAMIDE MALEATE Suppliers
Global( 33)Suppliers
Supplier | Tel | Country | ProdList | Advantage | Inquiry |
---|---|---|---|---|---|
TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 | United States | 19892 | 58 | Inquiry |
Aladdin Scientific | +1-+1(833)-552-7181 | United States | 52927 | 58 | Inquiry |
Amadis Chemical Company Limited | 571-89925085 | China | 131980 | 58 | Inquiry |
MedChemExpress | 021-58955995 | United States | 6398 | 58 | Inquiry |
United States Biological | 800.520.3011 or 781.639.5092 | United States | 6256 | 80 | Inquiry |
Jiangsu Aikon Biopharmaceutical R&D co.,Ltd. | 025-66099280 17798518460 | China | 19918 | 55 | Inquiry |
MedBioPharmaceutical Technology Inc | 021-69568360 18916172912 | China | 8141 | 58 | Inquiry |
Shanghai Universal Biotech Co.,Ltd | 18768175414 | China | 24998 | 58 | Inquiry |
Beijing Jin Ming Biotechnology Co., Ltd. | 010-60605840 15801484223; | China | 29778 | 58 | Inquiry |
TargetMol Chemicals Inc. | 4008200310 | China | 23963 | 58 | Inquiry |
106243-16-7(THIOPERAMIDE MALEATE)Related Search:
N-CYCLOHEXYL-4-(1H-IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
MR 12842
THIOPERAMIDE MALEATE
THIOPERAMIDE MALEATE SALT
THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE
N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide
Thiop
N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide
thioperamide
N-CYCLOHEXYL-4-(IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE
N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
1-Piperidinecarbothioamide, N-cyclohexyl-4-(1H-imidazol-5-yl)-
106243-16-7
C15H24N4SC4H4O4
Potent and selective H3 histamine receptor antagonist that crosses the blood-brain barrier.
Histamine receptor
Histamine