THIOPERAMIDE MALEATE

THIOPERAMIDE MALEATE Structure
CAS No.
106243-16-7
Chemical Name:
THIOPERAMIDE MALEATE
Synonyms
Thiop;MR 12842;thioperamide;THIOPERAMIDE MALEATE;THIOPERAMIDE MALEATE SALT;THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE;N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide;N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide;N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE;N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
CBNumber:
CB5245732
Molecular Formula:
C15H24N4S
Molecular Weight:
292.44
MOL File:
106243-16-7.mol
MSDS File:
SDS
Modify Date:
2023/6/30 15:45:59

THIOPERAMIDE MALEATE Properties

storage temp. Store at -20°C
solubility H2O: 10 mg/mL
form solid
color white

SAFETY

Risk and Safety Statements

Hazard Codes  Xi
Risk Statements  36/37/38
Safety Statements  26-36
WGK Germany  3

THIOPERAMIDE MALEATE Chemical Properties,Uses,Production

Uses

Thioperamide is a highly potent and selective ligand for histamine H3-receptors.

Biological Activity

Potent histamine H 3 and H 4 antagonist/inverse agonist. K i values are 25 and 27 nM for human recombinant H 3 and H 4 receptors respectively. Blocks eosinophil shape change (IC 50 = 1.4 μ M) and chemotaxis (IC 50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H 3 Receptor Tocriset™ .

THIOPERAMIDE MALEATE Preparation Products And Raw materials

Raw materials

Preparation Products

THIOPERAMIDE MALEATE Suppliers

Global( 33)Suppliers
Supplier Tel Country ProdList Advantage Inquiry
TargetMol Chemicals Inc. +1-781-999-5354 +1-00000000000 United States 19892 58 Inquiry
Aladdin Scientific +1-+1(833)-552-7181 United States 52927 58 Inquiry
Amadis Chemical Company Limited 571-89925085 China 131980 58 Inquiry
MedChemExpress 021-58955995 United States 6398 58 Inquiry
United States Biological 800.520.3011 or 781.639.5092 United States 6256 80 Inquiry
Jiangsu Aikon Biopharmaceutical R&D co.,Ltd. 025-66099280 17798518460 China 19918 55 Inquiry
MedBioPharmaceutical Technology Inc 021-69568360 18916172912 China 8141 58 Inquiry
Shanghai Universal Biotech Co.,Ltd 18768175414 China 24998 58 Inquiry
Beijing Jin Ming Biotechnology Co., Ltd. 010-60605840 15801484223; China 29778 58 Inquiry
TargetMol Chemicals Inc. 4008200310 China 23963 58 Inquiry
N-CYCLOHEXYL-4-(1H-IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE MR 12842 THIOPERAMIDE MALEATE THIOPERAMIDE MALEATE SALT THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide Thiop N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide thioperamide N-CYCLOHEXYL-4-(IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide 1-Piperidinecarbothioamide, N-cyclohexyl-4-(1H-imidazol-5-yl)- 106243-16-7 C15H24N4SC4H4O4 Potent and selective H3 histamine receptor antagonist that crosses the blood-brain barrier. Histamine receptor Histamine