Chinese english Japanese Germany Korea

KETANSERIN TARTRATE

KETANSERIN TARTRATE Structure
CAS No.
83846-83-7
Chemical Name:
KETANSERIN TARTRATE
Synonyms
kjk-945;R 41468;R41468 tartrate;Ketanserin Tartrat;Ketanserinetartrate;KETANSERIN TARTRATE;R 41468 TARTRATE SALT;quinazoline-2,4(1H,3H);KETANSERIN TARTRATE SALT;3-(2-(4-(4-Fluorobenzoyl)
CBNumber:
CB8415888
Molecular Formula:
C26H28FN3O9
Molecular Weight:
545.52
MOL File:
83846-83-7.mol
MSDS File:
SDS
Modify Date:
2023/6/30 15:45:59
Request For Quotation

KETANSERIN TARTRATE Properties

Melting point 183～186℃
storage temp. 2-8°C
solubility ethanol: 3.3mg/mL
form solid
color white
Water Solubility Soluble to 10 mM in water
CAS DataBase Reference 83846-83-7(CAS DataBase Reference)

SAFETY

Risk and Safety Statements

Symbol(GHS) 
GHS06
Signal word  Danger
Hazard statements  H301
Precautionary statements  P301+P310
Hazard Codes  T
Risk Statements  25
Safety Statements  22-36/37/39-45
RIDADR  UN 2811 6.1/PG 3
WGK Germany  3
RTECS  VA1411195
HazardClass  6.1
HS Code  29335990
Toxicity LD50 oral in rat: 129mg/kg
NFPA 704
0
2 0

KETANSERIN TARTRATE price More Price(5)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Sigma-Aldrich(India) S006 Ketanserin (+)-tartrate salt ≥97%, solid 83846-83-7 10MG ₹8919.8 2022-06-14 Buy
Sigma-Aldrich(India) S006 Ketanserin (+)-tartrate salt ≥97%, solid 83846-83-7 50MG ₹25395.45 2022-06-14 Buy
Sigma-Aldrich(India) S006 Ketanserin (+)-tartrate salt ≥97%, solid 83846-83-7 250MG ₹73480.1 2022-06-14 Buy
Sigma-Aldrich(India) S006 Ketanserin (+)-tartrate salt ≥97%, solid 83846-83-7 500MG ₹128265.43 2022-06-14 Buy
Sigma-Aldrich(India) 5.06271 Ketanserin Tartrate - CAS 83846-83-7 - Calbiochem 83846-83-7 50MG ₹12940 2022-06-14 Buy
Product number Packaging Price Buy
S006 10MG ₹8919.8 Buy
S006 50MG ₹25395.45 Buy
S006 250MG ₹73480.1 Buy
S006 500MG ₹128265.43 Buy
5.06271 50MG ₹12940 Buy

KETANSERIN TARTRATE Chemical Properties,Uses,Production

Description

Ketanserin is a potent antagonist of the serotonin (5-HT) receptor that is selective for 5-HT2 (IC50 = 6.3 nM; Ki = 2.1 nM). It has no activity at 5-HT1 receptors but does have activity at histamine type 1, α1-adrenergic, and dopamine receptors with Ki values of 10, 10, and 220 nM, respectively. Ketanserin induces dose-dependent inhibition of contractile responses to 5-HT in isolated rat caudal artery, canine basilar, carotid, coronary and gastrosplenic arteries, and canine gastrosplenic and saphenous veins. Ketanserin (10 mg/kg/day) significantly decreases blood pressure (BP), blood pressure variability (BPV), and hypertensive organ damage in spontaneously hypertensive rats. Formulations containing ketanserin have been used to treat hypertension in early-onset preeclampsia.

Uses

coccidiostat

Biological Activity

Selective 5-HT 2A serotonin receptor antagonist; can also be used to discriminate between 5-HT 1D and 5-HT 1B receptor subtypes.

KETANSERIN TARTRATE Preparation Products And Raw materials

Raw materials

Preparation Products

KETANSERIN TARTRATE Suppliers

Global( 140)Suppliers
Supplier Tel Country ProdList Advantage Inquiry
A.J Chemicals 91-9810153283 New Delhi, India 6124 58 Inquiry
Henan Bao Enluo International TradeCo.，LTD +86-17331933971 +86-17331933971 China 2503 58 Inquiry
Shanghai Daken Advanced Materials Co.,Ltd +86-371-66670886 China 16209 58 Inquiry
career henan chemical co +86-0371-86658258 +8613203830695 China 29826 58 Inquiry
Zhengzhou Alfa Chemical Co.,Ltd +8618530059196 China 12997 58 Inquiry
SIMAGCHEM CORP +86-13806087780 China 17367 58 Inquiry
TargetMol Chemicals Inc. +1-781-999-5354 +1-00000000000 United States 19892 58 Inquiry
AFINE CHEMICALS LIMITED +86-0571-85134551 China 15395 58 Inquiry
Finetech Industry Limited +86-27-87465837 +8618971612321 China 9626 58 Inquiry
Wuhan Fortuna Chemical Co., Ltd +86-027-59207850 China 5963 58 Inquiry
Supplier Advantage
A.J Chemicals 58
Henan Bao Enluo International TradeCo.，LTD 58
Shanghai Daken Advanced Materials Co.,Ltd 58
career henan chemical co 58
Zhengzhou Alfa Chemical Co.,Ltd 58
SIMAGCHEM CORP 58
TargetMol Chemicals Inc. 58
AFINE CHEMICALS LIMITED 58
Finetech Industry Limited 58
Wuhan Fortuna Chemical Co., Ltd 58

83846-83-7(KETANSERIN TARTRATE)Related Search:

2-(4-BENZYLPIPERIDINO)-1-ETHANAMINE 4-BENZOYLPIPERIDINE HYDROCHLORIDE 4-(4'-Fluorobenzyl)piperidine Butanedioic acid,2,3-dihydroxy- (2R,3R)-, ammonium salt (1:) KETANSERIN TARTRATE
BENZOYLUREA 4-(4-Fluorobenzoyl)piperidine N-(2-Aminoethyl)piperidine 1-(4-FLUORO-PHENYL)-BUTAN-1-ONE Benzoyleneurea
Ketanserin 4'-Fluoropropiophenone 4-Benzylpiperidine 1-(4-FLUOROPHENYL)-2-METHYLPROPAN-1-ONE 5-Diethylamino-2-pentanone
CHEMBRDG-BB 4013122 3,4-DIHYDROQUINAZOLIN-2(1H)-ONE 3,4-DIHYDRO-3-METHYL-2(1H)-QUINAZOLINONE
chevron_left

1of4

chevron_right
R 41468 R 41468 TARTRATE SALT 3-(2-(4-(p-fluorobenzoyl)-1-piperidinyl)ethyl)-2,4(1h,3h)-quinazolinedionel 4(1h,3h)-quinazolinedione,3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-( kjk-945 r-(r*,r*))-2,3-dihydroxybutanedioate(1:1) 3-[2-[4-(4-fluorobenzoyl)piperidino]ethyl]quinazoline-2,4(1H,3H)-dione [R-(R*,R*)]-tartrate KETANSERIN TARTRATE (R 41468) (SELECTIVE 5-HT2/5-HT1C SEROTONI Ketanserinetartrate R 41468 (+)-tartrate salt, 3-(2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl)-2,4(1H,3H)-quinazolinedione (+)-tartrate salt 3-[2-[4-(4-Fluorobenzoyl)piperidino]ethyl]-2,4-(1H,3H)-quinazolinedione tartrate Ketanserin Tartrat 3-(2-(4-(4-fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione 2,3-dihydroxysuccinate 3-(2-(4-(4-Fluorobenzoyl) -dione 2,3-dihydroxysuccinate quinazoline-2,4(1H,3H) Ketanserin tartrate salt Morpholino 3-[2-(4-FLUOROBENZOYL)-1-PIPERDINYL]-ETHYL]-2,4(1H,3H)-QUINAZOLINEDIONE TARTRATE 3-[2-[4-(4-FLUOROBENZOYL)-1-PIPERDINYL]ETHYL]-2,4(1H,3H)-QUINAZOLINEDIONE 3-[2-[4-(4-FLUOROBENZOYL)-1-PIPERDINYL]ETHYL]-2,4(1H,3H)-QUINAZOLINEDIONE TARTRATE 3-[2-[4-(4-FLUOROBENZOYL)-1-PIPERIDINYL]ETHYL]-2,4[1H,3H]-QUINAZOLINEDIONE TARTRATE 3-(2-[4-(4-FLUOROBENZOYL)-1-PIPERIDINYL]ETHYL)-2,4(1H,3H)-QUINAZOLINEDIONE TARTRATE SALT KETANSERIN TARTRATE KETANSERIN TARTRATE SALT R41468 tartrate 3-[2-[4-[(4-fluorophenyl)-oxomethyl]-1-piperidin-1-iumyl]ethyl]-1H-quinazoline-2,4-dione Ketanserin tartrate (R41468 tartrate) Ketanserin Tartrate - CAS 83846-83-7 - Calbiochem Ketanserin Hydrogen Tartrate 2,4(1H,3H)-Quinazolinedione,3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-,(2R,3R)-2,3-dihydroxybutanedioate (1:1) 3-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione (2R,3R)-2,3-dihydroxysuccinate 83846-83-7 C22H22FN3O3C4H6O6 C26H28N3O9F C4H6O6C22H22FN3O3 C26H28FN3O9 Biochemicals and Reagents Enzyme Inhibitors Other Enzymes, Inhibitors, and Substrates Enzyme Inhibitors by Type BioChemical Serotonin Cardiovascular APIs Serotonin receptor