SB 269970 HYDROCHLORIDE 化学特性,用途語,生産方法
使用
SB 269970 is a selective and potent SR-7 antagonist.
生物活性
Potent and selective 5-HT 7 receptor antagonist (pK i values are 8.9, 7.2 and 6.0 for 5-HT 7A , 5-HT 5A and 5-HT 1B and < 6.0 for 5-HT 1A , 5-HT 1D , 5-HT 1E , 5-HT 1F , 5-HT 2A , 5-HT 2B , 5-HT 2C , 5-HT 4 and 5-HT 6 receptors respectively). Brain penetrant in vivo .
SB 269970 HYDROCHLORIDE 上流と下流の製品情報
原材料
準備製品