クエン酸スフェンタニル

クエン酸スフェンタニル 化学特性,用途語,生産方法

効能

麻薬性鎮痛薬, オピオイド受容体作動薬

化学的特性

Crystalline Solid

使用

Potent derivative of Fentanyl. Analgesic (narcotic). Controlled substance (opiate)

一般的な説明

Sufentanil is a short acting synthetic opioid analgesic most commonly used for pain relief during medical operations. This certified solution standard is applicable to use in clinical toxicology, pain prescription monitoring, or forensic analysis by LC-MS/MS or GC/MS. Sufentanil is sold under the trade name Sufenta.

臨床応用

Addition of the 4-methoxymethyl group and bioisosteric replacement of the phenyl with a 2-thiophenyl on the fentanyl structure results in a 10-fold increase in μ opioid activity. The resultant compound, sufentanil, is 600 to 800 times more potent than morphine. Despite its greater sedative and analgesic potency, sufentanil produces less respiratory depression at effective anesthetic doses. Sufentanil is available in an intravenous dosage form, and it is used for anesthetic procedures. It has a faster onset and shorter duration of action than fentanyl. The short duration is caused by redistribution from brain tissues after intravenous dosage.

クエン酸スフェンタニル 上流と下流の製品情報

原材料

準備製品

60561-17-3(クエン酸スフェンタニル)キーワード:

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• 60561-17-3
• SUFENTANIL CITRATE
• n-(4-(methoxymethyl)-1-(2-(2-thienyl)ethyl)-4-piperidinyl)-n-phenylpropionam
• n-(4-(methoxymethyl)-1-(2-(2-thienyl)ethyl)-4-piperidyl)-propionanilidcitr
• n-(4-(methoxymethyl)-1-(2-(2-thienyl)ethyl)-4-piperidyl)propionanilidecitrat
• r30730citratesalt
• r33800
• sufentanylcitrate
• N-[4-(methoxymethyl)-1-[2-(2-thienyl)ethyl]-4-piperidyl]-N-phenylpropionamide citrate
• SUFENTANILCITRATE,USP
• Propanamide, N-[4-(methoxymethyl)-1-[2- (2-thienyl)ethyl]-4-piperidinyl]-N-phenyl-, 2-hydroxy-1,2,3-propanetricarboxylate (1:1)
• N-[4-(Methoxymethyl)-1-[2-(2-thienyl)ethyl]-4-piperidinyl]-N-phenyl, propanamide 2-Hydroxy-1,2,3-propanetricarboxylate
• Sufenta
• Sufentanil Forte
• Sufentanyl Citrat
• Sufentanil Citrate CII (25 mg)
• Methanol（Test:Sufentanil Citrate, 100 μg/mL as free base）
• Sufentanil Citrate (CII), USP
• Sufentanil Citrate solution
• N-[4-(Methoxymethyl)-1-[2-(2-thienyl)ethyl]-4-piperidinyl]-N-phenylpropanamide citrate
• Sufentanil Citrate CII (1623648)
• Sufentanil citrate salt
• OJCZPLDERGDQRJ-UHFFFAOYSA-N
• Rezvilutamide Impurity 38
• N-[4-メトキシメチル-1-[2-(2-チエニル)エチル]-4-ピペリジニル]-N-フェニルプロパンアミド·2-ヒドロキシ-1,2,3-プロパントリカルボン酸
• スフェンタニルくえん酸塩
• N-[4-(メトキシメチル)-1-[2-(2-チエニル)エチル]-4-ピペリジニル]-N-フェニルプロパンアミド·2-ヒドロキシ-1,2,3-プロパントリカルボン酸
• くえん酸スフェンタニル
• スフェンタニルシトラート