RO-31-8220 化学特性,用途語,生産方法
使用
Ro 31-8220 Mesylate is a protein kinase C (PKC) inhibitor.
一般的な説明
Ro 31-8220 is a bisindolylmaleimide derivative of staurosporine. Ro 31-8220 blocks MAP kinase phosphatase-1 (MKP-1) expression, induces c-Jun expression and stimulates Jun N-terminal Kinase (JNK1). It has immunosuppressive properties.
Biochem/physiol Actions
Inhibitor of GRK-5 (G protein-coupled receptor kinase); PKC (protein kinase C); MAPKAP kinase 1β and p70 S6 kinase.
RO-31-8220 上流と下流の製品情報
原材料
準備製品