BQ-788
- $175 - $5000
- Product name: BQ-788
- CAS: 156161-89-6
- MF: C34H52N5NaO7
- MW: 665.81
- EINECS:
- MDL Number:MFCD00797882
- Synonyms:BQ-788 SODIUM;BQ-788 SYNTHETIC >97% ETB ENDOTHELIN REC EPT;N-[(cis-2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucinesodiumsalt;1-ELAIDYLPHOSPHOCHOLINE, >97%;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl]-1-(methoxycarbonyl)-D-tryptophyl]-D-norleucine sodium salt, 2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-;DMpc-gaMMa-MeLeu-D-Trp(1-CO2CH3)-D-Nle.Na (DMpc : cis-2,6-DiMethylpiperidinocarbonyl);2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
15 prices
Selected condition:
Brand
- Adipogen Life Sciences
- AK Scientific
- Alichem
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Sigma-Aldrich
- TRC
Package
- 200μg
- 500μg
- 1mg
- 5mg
- 10mg
- 100mg
- 250mg
- 1g
- ManufacturerAdipogen Life Sciences
- Product numberAG-CP3-0012-M001
- Product descriptionBQ-788.sodiumsalt ≥95%(HPLC)
- Packaging1mg
- Price$200
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number3506AH
- Product descriptionDMPC-Gamma-MELEU-D-Trp(1-Co2CH3)-D-NleNa
- Packaging1mg
- Price$368
- Updated2021-12-16
- Buy
- ManufacturerAlichem
- Product number156161896
- Product descriptionSodiumBQ-788
- Packaging10mg
- Price$400
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number17403
- Product descriptionBQ-788 (sodium salt) ≥95%
- Packaging500μg
- Price$175
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number17403
- Product descriptionBQ-788 (sodium salt) ≥95%
- Packaging1mg
- Price$242
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-2685
- Product descriptionBQ-788(sodiumsalt) 98.03%
- Packaging1mg
- Price$180
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-2685
- Product descriptionBQ-788(sodiumsalt) 98.03%
- Packaging5mg
- Price$420
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-2685
- Product descriptionBQ-788(sodiumsalt) 98.03%
- Packaging10mg
- Price$600
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31003231
- Product descriptionSodiumBQ-788 98+%
- Packaging5mg
- Price$345
- Updated2021-12-16
- Buy
- ManufacturerCSNpharm
- Product numberCSN17348
- Product descriptionBQ-788Sodium
- Packaging5mg
- Price$336
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7542
- Product descriptionBQ-788 >98%
- Packaging100mg
- Price$1250
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7542
- Product descriptionBQ-788 >98%
- Packaging250mg
- Price$2500
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7542
- Product descriptionBQ-788 >98%
- Packaging1g
- Price$5000
- Updated2021-12-16
- Buy
- ManufacturerSigma-Aldrich
- Product numberB157
- Product descriptionBQ-788 ≥95%,solid
- Packaging200μg
- Price$231
- Updated2024-03-01
- Buy
- ManufacturerTRC
- Product numberB676670
- Product descriptionBQ788
- Packaging5mg
- Price$595
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
Adipogen Life Sciences | AG-CP3-0012-M001 | BQ-788.sodiumsalt ≥95%(HPLC) | 1mg | $200 | 2021-12-16 | Buy |
AK Scientific | 3506AH | DMPC-Gamma-MELEU-D-Trp(1-Co2CH3)-D-NleNa | 1mg | $368 | 2021-12-16 | Buy |
Alichem | 156161896 | SodiumBQ-788 | 10mg | $400 | 2021-12-16 | Buy |
Cayman Chemical | 17403 | BQ-788 (sodium salt) ≥95% | 500μg | $175 | 2024-03-01 | Buy |
Cayman Chemical | 17403 | BQ-788 (sodium salt) ≥95% | 1mg | $242 | 2024-03-01 | Buy |
ChemScene | CS-2685 | BQ-788(sodiumsalt) 98.03% | 1mg | $180 | 2021-12-16 | Buy |
ChemScene | CS-2685 | BQ-788(sodiumsalt) 98.03% | 5mg | $420 | 2021-12-16 | Buy |
ChemScene | CS-2685 | BQ-788(sodiumsalt) 98.03% | 10mg | $600 | 2021-12-16 | Buy |
Crysdot | CD31003231 | SodiumBQ-788 98+% | 5mg | $345 | 2021-12-16 | Buy |
CSNpharm | CSN17348 | BQ-788Sodium | 5mg | $336 | 2021-12-16 | Buy |
DC Chemicals | DC7542 | BQ-788 >98% | 100mg | $1250 | 2021-12-16 | Buy |
DC Chemicals | DC7542 | BQ-788 >98% | 250mg | $2500 | 2021-12-16 | Buy |
DC Chemicals | DC7542 | BQ-788 >98% | 1g | $5000 | 2021-12-16 | Buy |
Sigma-Aldrich | B157 | BQ-788 ≥95%,solid | 200μg | $231 | 2024-03-01 | Buy |
TRC | B676670 | BQ788 | 5mg | $595 | 2021-12-16 | Buy |
Properties
storage temp. :-20°C
solubility :acetonitrile: 0.3 mg/mL
form :solid
color :white
solubility :acetonitrile: 0.3 mg/mL
form :solid
color :white
Safety Information
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Description
The endothelin (ET) family of proteins mediate a variety of responses, with ET-1 being a potent and long-lasting constrictor of human cardiovascular vessels. These proteins activate the G protein-coupled receptors ETA and ETB, with ETB being non-specific for ET protein form. BQ-788 is a potent, selective antagonist of ETB (IC50 = 1.2 nM for blocking ET-1 binding to human Girardi heart cells). It weakly inhibits the binding of ET-1 to ETA receptors on human neuroblastoma SK-N-MC cells (IC50 = 1300 nM). BQ-788 competitively antagonizes the vasoconstriction induced by an ETB-selective agonist on isolated rabbit pulmonary arteries, blocks ET-1 induced bronchoconstriction in guinea pigs, and abolishes an ET-1 mediated depressor response in rats.Related product price
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