Company Name: |
ATK CHEMICAL COMPANY LIMITED
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Tel: |
+undefined-21-51877795 |
Email: |
ivan@atkchemical.com |
Products Intro: |
Product Name:IRL 2500 CAS:169545-27-1 Purity:98% Package:10MG;50MG;100MG,1G,5G,10G
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Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
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Tel: |
821-50328103-801 18930552037 |
Email: |
3bsc@sina.com |
Products Intro: |
Product Name:IRL-2500;N-3-[1,1'-Biphenyl]-4-yl-N-(3,5-diMethylbenzoyl)-N-Methyl-D-alanyl-L-tryptophan CAS:169545-27-1 Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
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| IRL-2500 Basic information |
Product Name: | IRL-2500 | Synonyms: | IRL-2500;N-3-[1,1'-BIPHENYL]-4-YL-N-(3,5-DIMETHYLBENZOYL)-N-METHYL-D-ALANYL-L-TRYPTOPHAN;((R)-3-([1,1'-Biphenyl]-4-yl)-2-(N,3,5-trimethylbenzamido)propanoyl)-L-tryptophan;L-Tryptophan, 3-[1,1'-biphenyl]-4-yl-N-(3,5-dimethylbenzoyl)-N-methyl-D-alanyl-;((R)-3-([1,1'-Biphenyl]-4-yl)-2-(N,3,5-trimethylbenzamido)propanoyl)-L-tryptophan | CAS: | 169545-27-1 | MF: | C36H35N3O4 | MW: | 573.68 | EINECS: | | Product Categories: | Endothelin receptor | Mol File: | 169545-27-1.mol | |
| IRL-2500 Chemical Properties |
Boiling point | 893.7±65.0 °C(Predicted) | density | 1.246±0.06 g/cm3(Predicted) | storage temp. | Keep in dark place,Sealed in dry,Store in freezer, under -20°C | solubility | Soluble to 100 mM in 1eq. NaOH | form | Powder | pka | 3.34±0.10(Predicted) | color | White to light yellow |
| IRL-2500 Usage And Synthesis |
Uses | IRL 2500 is a potent endothelin ETB selective antagonist. | Biological Activity | Potent endothelin receptor antagonist; shows some selectivity for ET B receptors (IC 50 values are 1.3 and 94 nM for ET B and ET A receptors respectively). Inhibits ET B receptor-mediated blood pressure increase and renal vascular resistance in rats in vivo . | storage | Desiccate at RT |
| IRL-2500 Preparation Products And Raw materials |
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