中文名:阿塞那平盐酸盐
英文名:Asenapine maleate
中文别名:阿塞那平马来酸盐|马来酸阿塞那平
英文别名:Asenapine maleate|85650-56-2|Saphris|Asenapine (maleate)|Org 5222|Org-5222|Sycrest|Asenapine maleate [USAN]|UNII-CU9463U2E2|Asenapine (as maleate)|CU9463U2E2|EINECS 288-064-8|(Z)-but-2-enedioic acid;(2S,6S)-9-chloro-4-methyl-13-oxa-4-azatetracyclo[12.4.0.
纯度:≥98% (HPLC)
货号:A124739
包装:10mg、50mg、250mg
Cas号:85650-56-2
存储温度:2-8°C储存
产品介绍:
Asenapine maleate是 5-HT(1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和 D2 的拮抗剂,Ki 值分别为 0.03-4.0 nM, 1.3 nM。同时也是一种抗精神病药物。Asenapine maleate has been used as a stressor in studying the Fos expression in forebrain structures of rat models. Asenapine maleate is a serotonin 5-HT and dopamine D2 receptor antagonist. Asenapine maleate can be used to treat schizophrenia and bipolar mania.
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