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Muscarinic toxin 1

 структура
CAS №
английское имя:
Muscarinic toxin 1
Синонимы:
MT1;MTX1;MEL-1A-R;MT1; MT 1;MUSCARINIC TOXIN 1;Mel1a melatonin receptor;Anti-MTR1A antibody produced in rabbit;Anti-MTNR1A antibody produced in rabbit;Muscarinic Toxin-1 from Dendroaspis angusticeps venom;LEU-THR-CYS-VAL-THR-SER-LYS-SER-ILE-PHE-GLY-ILE-THR-THR-GLU-ASN-CYS-PRO-ASP-GLY-GLN-ASN-LEU-CYS-PHE-LYS-LYS-TRP-TYR-TYR-ILE-VAL-PRO-ARG-TYR-SER-ASP-ILE-THR-TRP-GLY-CYS-ALA-ALA-THR-CYS-PRO-LYS-PRO-THR-ASN-VAL-ARG-GLU-THR-ILE-ARG-CYS-CYS-GLU-THR-ASP-LYS-CYS-ASN-GLU
CBNumber:
CB3392337
Формула:
молекулярный вес:
0
MOL File:
Mol file

Muscarinic toxin 1 атрибут

температура хранения: −20°C
форма: лиофилизированный порошок

Заявления о рисках и безопасности

WGK Германия 3

Muscarinic toxin 1 химические свойства, назначение, производство

Биологические функции

Muscarinic toxin 1 has non-competitive interactions with adrenergic and muscarinic receptors. Binds to alpha-2b (ADRA2B) (IC50=2.3 nM), alpha-1a (ADRA1A), alpha-1b (ADRA1B) and alpha-2c (ADRA2C) adrenergic receptors. Reversibly binds to the M1 (CHRM1) muscarinic acetylcholine receptor, probably through interaction with the orthosteric site. Also has slightly weaker effects on M3 (CHRM3) and M4 (CHRM4) receptors. The order of potency is ADRA2B>>CHRM1>ADRA1A>ADRA1B>ADRA2C/CHRM4 (PubMed:24793485).

Muscarinic toxin 1 препаратная продукция и сырье

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препарат


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