PNU 37883 hydrochloride химические свойства, назначение, производство
Биологическая активность
Novel antagonist selective for the vascular form of K ATP channel; inhibits K ATP currents in isolated mesenteric artery smooth muscle cells (K d = 65 nM) but not in cardiac or skeletal myocytes. In vivo, inhibits blood vessel relaxation and hypotension induced by pinacidil. Displays weak diuretic effects.
PNU 37883 hydrochloride препаратная продукция и сырье
сырьё
препарат