SHU-9119
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- $77 - $3300
- Product name: SHU-9119
- CAS: 168482-23-3
- MF: C54H71N15O9
- MW: 1074.24
- EINECS:
- MDL Number:MFCD01631255
- Synonyms:SHU-9119;[N-ACETYL-NLE4,ASP5,D-2'-NAL7,LYS10]-ALPHA-MSH (4-10) AMIDE, ASP5-LYS10, CYCLIC LACTAM;AC-NLE-ASP-HIS-D-2-NAL-ARG-TRP-LYS-NH2;AC-NLE-ASP-HIS-D-2'-NAL-ARG-TRP-LYS-NH2, ASP5-LYS10, CYCLIC LACTAM;AC-NLE-ASP-HIS-D-2-NAL-H2N-LYS-TRP-ARG;AC-NLE-ASP-HIS-D-NAL(2)-ARG-TRP-LYS-NH2;(AC-NLE4,ASP5,D-2-NAL7,LYS10)-CYCLO-ALPHA-MSH (4-10) AMIDE;AC-[NLE4, ASP5, D-2-NAL7, LYS10]-CYCLO-ALPHA-MSH AMIDE (4-10)
12 prices
Selected condition：
Brand
- American Custom Chemicals Corporation
- ApexBio Technology
- Cayman Chemical
- ChemScene
- DC Chemicals
- Tocris
- Usbiological
Package
- 1
- 500μg
- 1MG
- 5MG
- 100mg
- 1g
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberPEP0003113
- Product descriptionSHU 9119 95.00%
- Packaging1MG
- Price$643.98
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberPEP0003113
- Product descriptionSHU 9119 95.00%
- Packaging5MG
- Price$988.45
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB5425
- Product descriptionSHU9119
- Packaging1mg
- Price$173
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB5425
- Product descriptionSHU9119
- Packaging5mg
- Price$693
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number24152
- Product descriptionSHU9119 (trifluoroacetate salt) ≥95%
- Packaging500μg
- Price$77
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number24152
- Product descriptionSHU9119 (trifluoroacetate salt) ≥95%
- Packaging1mg
- Price$121
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-6496
- Product descriptionSHU9119 98.21%
- Packaging1mg
- Price$108
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6496
- Product descriptionSHU9119 98.21%
- Packaging5mg
- Price$468
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC22894
- Product descriptionSHU-9119 >98%
- Packaging1g
- Price$3300
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC22894
- Product descriptionSHU-9119 >98%
- Packaging100mg
- Price$900
- Updated2021-12-16
- Buy
- ManufacturerTocris
- Product number3420
- Product descriptionSHU9119
- Packaging1
- Price$151
- Updated2021-12-16
- Buy
- ManufacturerUsbiological
- Product number256659
- Product descriptionSHU 9119
- Packaging1mg
- Price$389
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| American Custom Chemicals Corporation | PEP0003113 | SHU 9119 95.00% | 1MG | $643.98 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | PEP0003113 | SHU 9119 95.00% | 5MG | $988.45 | 2021-12-16 | Buy |
| ApexBio Technology | B5425 | SHU9119 | 1mg | $173 | 2021-12-16 | Buy |
| ApexBio Technology | B5425 | SHU9119 | 5mg | $693 | 2021-12-16 | Buy |
| Cayman Chemical | 24152 | SHU9119 (trifluoroacetate salt) ≥95% | 500μg | $77 | 2024-03-01 | Buy |
| Cayman Chemical | 24152 | SHU9119 (trifluoroacetate salt) ≥95% | 1mg | $121 | 2024-03-01 | Buy |
| ChemScene | CS-6496 | SHU9119 98.21% | 1mg | $108 | 2021-12-16 | Buy |
| ChemScene | CS-6496 | SHU9119 98.21% | 5mg | $468 | 2021-12-16 | Buy |
| DC Chemicals | DC22894 | SHU-9119 >98% | 1g | $3300 | 2021-12-16 | Buy |
| DC Chemicals | DC22894 | SHU-9119 >98% | 100mg | $900 | 2021-12-16 | Buy |
| Tocris | 3420 | SHU9119 | 1 | $151 | 2021-12-16 | Buy |
| Usbiological | 256659 | SHU 9119 | 1mg | $389 | 2021-12-16 | Buy |
Properties
Density :1.43±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :H2O : 20 mg/mL (18.62 mM; Need ultrasonic)
form :Powder
pka :13.00±0.70(Predicted)
color :White to off-white
Water Solubility :Soluble to 0.20 mg/ml in water
Sequence :Ac-Nle-Asp-His-D-Nal-Arg-Trp-Lys-NH2(Chemical Bridge Asp2-Lys7)
storage temp. :-20°C
solubility :H2O : 20 mg/mL (18.62 mM; Need ultrasonic)
form :Powder
pka :13.00±0.70(Predicted)
color :White to off-white
Water Solubility :Soluble to 0.20 mg/ml in water
Sequence :Ac-Nle-Asp-His-D-Nal-Arg-Trp-Lys-NH2(Chemical Bridge Asp2-Lys7)
Safety Information
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Description
SHU9119 is an agonist of melanocortin receptor 1 (MC1R) and antagonist of MC4R (IC50s = 1.2 and 2.9 nM, respectively, for displacement of melanocortin). It induces cAMP formation in HEK293 cells expressing human MC1R (EC50 = 1.11 nM), but inhibits cAMP formation in cells expressing human MC4R. In rats, SHU9119 (24 nmol, i.c.v. per day for seven days) increases food intake, body weight, fat mass, and lean mass, with concomitant increases in blood glucose, insulin, and leptin levels via disrupted melanocortin signaling. Similarly, mice treated with SHU9119 (5 nmol/day, i.c.v.) exhibit food intake-independent increases in body weight and fat mass consequent to MC4R inhibition and subsequent brown adipose tissue dysfunction.More related product prices
Melanotan IIRelated product price
- Melanotan II
$35-3154.84 - SHU-9119
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$50-894