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JTC 801

JTC 801 Structure
CAS No.
244218-51-7
Chemical Name:
JTC 801
Synonyms
CS-161;JTC 801;JTC 801 HCl;JTC-801/JTC801;JTC 801 USP/EP/BP;JTC-801 >=98% (HPLC);JTC-801 hydrochloride;N-(4-Amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]benzamidehydrochloride;N-(4-AMino-2-Methyl-quinolin-6-yl)-2-(4-ethyl-phenoxyMethyl)-benzaMide hydrochloride;Benzamide,N-(4-amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]-, hydrochloride
CBNumber:
CB9812002
Molecular Formula:
C26H25N3O2.ClH
Molecular Weight:
447.963
MOL File:
244218-51-7.mol
MSDS File:
SDS
Modify Date:
2023/6/30 15:45:59

JTC 801 Properties

Melting point 235℃
storage temp. Inert atmosphere,2-8°C
solubility DMSO: ≥20mg/mL
form powder
color tan
InChIKey NQLIYKXNAXKMBL-UHFFFAOYSA-N

SAFETY

Risk and Safety Statements

Symbol(GHS) 
GHS07
Signal word  Warning
Hazard statements  H319
Precautionary statements  P264-P280-P305+P351+P338-P337+P313
Hazard Codes  Xi
Risk Statements  36
Safety Statements  26
WGK Germany  1
NFPA 704
0
2 0

JTC 801 price More Price(2)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Sigma-Aldrich(India) J3955 JTC-801 ≥98% (HPLC) 244218-51-7 5MG ₹14927.68 2022-06-14 Buy
Sigma-Aldrich(India) J3955 JTC-801 ≥98% (HPLC) 244218-51-7 25MG ₹60187 2022-06-14 Buy
Product number Packaging Price Buy
J3955 5MG ₹14927.68 Buy
J3955 25MG ₹60187 Buy

JTC 801 Chemical Properties,Uses,Production

Uses

JTC 801 is a novel opioid receptor-like1 (ORL1) receptor antagonist.

Biological Activity

High affinity, selective NOP receptor antagonist (K i = 8.2 nM). Displays approximately 12.5-, 129- and 1055-fold selectivity over human μ -, κ - and δ -opioid receptors respectively. In vivo shows anti-nociceptive effects in acute pain models. Orally active.

JTC 801 Preparation Products And Raw materials

Raw materials

Preparation Products

Global( 109)Suppliers
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ATK CHEMICAL COMPANY LIMITED +undefined-21-51877795 China 32760 60 Inquiry
CONIER CHEM AND PHARMA LIMITED +8618523575427 China 49391 58 Inquiry
career henan chemical co +86-0371-86658258 +8613203830695 China 29825 58 Inquiry
Dideu Industries Group Limited +86-29-89586680 +86-15129568250 China 24330 58 Inquiry
Zhejiang J&C Biological Technology Co.,Limited +1-2135480471 +1-2135480471 China 10522 58 Inquiry
Labnetwork lnc. +86-27-50766799 +8618062016861 China 19994 58 Inquiry
InvivoChem +1-708-310-1919 +1-13798911105 United States 6393 58 Inquiry
LEAP CHEM CO., LTD. +86-852-30606658 China 24738 58 Inquiry
Coresyn Pharmatech Co., Ltd. +86-571-86626709 +86-18157142896 China 9991 58 Inquiry
TargetMol Chemicals Inc. +1-781-999-5354 United States 19973 58 Inquiry
JTC 801 N-(4-Amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]benzamidehydrochloride N-(4-Amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]benzamide monohydrochloride JTC 801 HCl JTC-801 hydrochloride JTC-801/JTC801 N-(4-AMino-2-Methyl-quinolin-6-yl)-2-(4-ethyl-phenoxyMethyl)-benzaMide hydrochloride Benzamide,N-(4-amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]-, hydrochloride CS-161 JTC-801 >=98% (HPLC) JTC 801 USP/EP/BP 244218-51-7 Inhibitors