SクリPテイド 化学特性,用途語,生産方法
説明
Scriptaid is a histone deacetylase inhibitor that has an optimal concentration of 6-
8 μM in a cell-
based assay, is less toxic than trichostatin A, and works in a wide variety of biological systems. It induces cell cycle arrest in colon cancer cells in culture and inhibits tumor growth
in vitro and
in vivo. Scriptaid also facilitates the cloning of inbred mouse strains produced by somatic cell nuclear transfer.
使用
Scriptaid has been used in post activation of oocytes and embryo culture.
一般的な説明
Scriptaid is a histone deacetylase (HDAC) inhibitor, which enhances global acetylation of histones. It improves transcriptional activity and protein expression. Scriptaid inhibits tumor growth. It decreases telomerase activity and stimulates glioma cell apoptosis.
生物活性
Novel histone deacetylase inhibitor. Produces > 100-fold increase in histone acetylation and displays relatively low toxicity.
SクリPテイド 上流と下流の製品情報
原材料
準備製品