PROTAC ER Degrader-4

PROTAC ER Degrader-4 Suppliers list
Company Name: TargetMol Chemicals Inc.
Tel: +1-781-999-5354 +1-00000000000
Email: marketing@targetmol.com
Products Intro: Product Name:PROTAC ER Degrader-4
CAS:2361114-15-8
Purity:98.00% Package:100 mg;500 mg Remarks:REAGENT;FOR LABORATORY USE ONLY
Company Name: Sichuan Wei Keqi Biological Technology Co., Ltd.  
Tel: 028-81700200 18116577057
Email: 3003855609@qq.com
Products Intro: Product Name:PROTACERDegrader-4
CAS:2361114-15-8
Purity:98% Package:5mg;10mg;20mg;50mg;100mg;200mg;500mg;1g
Company Name: Shanghai Chaolan Chemical Technology Center  
Tel: QQ:65489617 15618227136
Email: info@SuperLan-chem.com
Products Intro: Product Name:PROTAC ER Degrader-4
CAS:2361114-15-8
Purity:98% HPLC Package:5MG;10MG;50MG;100MG,1G,5G,500G
Company Name: Jilin Province Woda Biotechnology Co., Ltd.  
Tel: 13504435624
Email: 1927928688@qq.com
Products Intro: Product Name:PROTAC ER Degrader-4
CAS:2361114-15-8
Purity:99% HPLC Package:1克;5克;
Company Name: Changzhou Bojia Biomedical Technology Co., Ltd.  
Tel: 2122619822
Email: czbjpharma@126.com
Products Intro: Product Name:PROTAC ER Degrader-4
CAS:2361114-15-8
Purity:99% Package:1g/10g/100g/1kg
PROTAC ER Degrader-4 Basic information
Product Name:PROTAC ER Degrader-4
Synonyms:PROTAC ER Degrader-4
CAS:2361114-15-8
MF:C53H67F3N6O8S
MW:1005.19
EINECS:
Product Categories:
Mol File:Mol File
PROTAC ER Degrader-4 Structure
PROTAC ER Degrader-4 Chemical Properties
Boiling point 1038.9±65.0 °C(Predicted)
density 1.254±0.06 g/cm3(Predicted)
pka13.54±0.46(Predicted)
form Solid
color Light yellow to yellow
Safety Information
MSDS Information
PROTAC ER Degrader-4 Usage And Synthesis
Biological ActivityPROTAC ER Degrader-4 is a von Hippel-Lindau-based PROATC estrogen receptor (ER) degrader, binding to ER with an IC50 of 0.8 nM. PROTAC ER Degrader-4 induces ER degradation in MCF-7 cells with an IC50 of 0.3 nM[1]. PROTAC ER Degrader-4 shows equal to 100% ER degradation at 0.3 μM in the MCF-7 ER degradation cellular assay[1].
References[1]. Bin Yang, et al. Compounds and their use in treating cancer. WO2019123367A1.
PROTAC ER Degrader-4 Preparation Products And Raw materials
Tag:PROTAC ER Degrader-4(2361114-15-8) Related Product Information
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