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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
4-[(S)-hydroxy-[(1S,2R,4S,5R)-5-vinylquinuclidin-2-yl]methyl]quinolin-6-ol (9S)- CINCHONAN-6',9-DIOL 70877-75-7 详细
4-[(2R)-2-(4-chloro-2-fluoro-phenyl)-2-methyl-1,3-benzodioxol-4-yl]piperidine;4-methylbenzenesulfonic acid 4-甲基苯磺酸 2832230-22-3 详细
tert-butyl 3-(aminomethyl)-3-pyrazol-1-yl-azetidine-1-carboxylate 2551119-71-0 详细
(6-diphenylphosphanyl-10H-phenoxazin-4-yl)-diphenyl-phosphane 4,6-二(二苯基膦)吩嗪 261733-18-0 详细
2-methoxy-4-(4-methylpiperazin-1-yl)aniline 2-甲氧基-4-(4-甲基哌嗪-1-基)苯胺 122833-04-9 详细
2-phenyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2-苯基-5-吡啶硼酸酯 879291-27-7 详细
1-methyl-3-phenyl-4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole 1-甲基-3-苯基-4-(4,4,5,5-四甲基-1,3,2-二恶硼烷-2-基)-1H-吡唑 1002334-06-6 详细
5-cyclopropyl-1h-pyrrolo[2,3-b]pyridine 5-环丙基-1h-吡咯并[2,3-b]吡啶 1254567-75-3 详细
4,4,5,5-tetramethyl-2-[(1S,2S)-2-phenylcyclopropyl]-1,3,2-dioxaborolane 4,4,5,5-四甲基-2-[((1S,2S)-2-苯基环丙基]-1,3,2-二氧杂硼烷 1240492-43-6 详细
tert-butyl (3R)-3-(oxetan-3-ylamino)piperidine-1-carboxylate 1349699-81-5 1349699-81-5 详细
(2R,3R)-3-(2,5-difluorophenyl)-3-hydroxy-2-methyl-4-(1H-1,2,4-triazol-1-yl)butanethioamide (2R,3R)-3-(2,5-二氟苯基)-3-羟基-2-甲基-4-(1H-1,2,4-三唑-1-基)丁烷硫代酰胺 368421-58-3 详细
(1S)-1-[4-methyl-5-[2-(trifluoromethyl)-4-pyridyl]-2-pyridyl]ethanamine (1S)-1-[4-甲基-2'-(三氟甲基)-[3,4'-联吡啶]-6-基]乙烷-1-胺 1628106-86-4 详细
fluoromethyl-phenyl-(2,3,4,5-tetramethylphenyl)sulfonium;tetrafluoroborate 四氟硼酸(氟甲基)(苯基)(2,3,4,5-四甲基苯基)硫鎓 1009088-40-7 详细
3-(5-amino-1-oxo-isoindolin-2-yl)piperidine-2,6-dione 来那度胺杂质13 191732-70-4 详细
tert-butyl 4-(6-chloro-2-pyridyl)piperidine-1-carboxylate 1-Piperidinecarboxylic acid, 4-(6-chloro-2-pyridinyl)-, 1,1-dimethylethyl ester 1266118-78-8 详细
Methanone, cyclopropylphenyl- 苯基环丙基甲酮 3481-02-5 详细
2-(2,6-dioxo-3-piperidyl)-5-iodo-isoindoline-1,3-dione 2-(2,6-二氧代哌啶-3-基)-5-碘异吲哚啉-1,3-二酮 2509137-01-1 详细
tert-butyl 3-(4-fluorophenyl)-3-(hydroxymethyl)azetidine-1-carboxylate 1-BOC-3-(4-氟苯基)-3-(羟甲基)氮杂环丁烷 2306262-31-5 详细
(2S)-oxiran-2-yl]methyl 3-nitrobenzene-1-sulfonate (S)-(+)-间硝基苯磺酸缩水甘油酯 115314-14-2 详细
(4R)-4-benzyl-3-propanoyl-1,3-oxazolidin-2-one (R)-(-)-4-苄基-3-丙酰基-2-恶唑烷酮 131685-53-5 详细
4-cyclohexylcyclohexan-1-ol 4-环已基环已醇 2433-14-9 详细
2-([1,1'-biphenyl]-3-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 3-联苯硼酸频呐醇酯 912844-88-3 详细
5-[(2R)-pyrrolidin-2-yl]-2H-1,2,3,4-tetrazole (R)-5-(吡咯烷-2-YL)-1H-四氮唑 702700-79-6 详细
tert-butyl 3-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]pyrrolidine-1-carboxylate 叔-丁基 3-[4-(四甲基-1,3,2-二噁硼戊环-2-基)-1H-吡唑-1-基]吡咯烷-1-甲酸基酯 1359974-18-7 详细
tert-butyl 4-{[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]methyl}piperidine-1-carboxylate 叔-丁基 4- 1092563-72-8 详细
tert-butyl 4-(aminomethyl)-4-phenylpiperidine-1-carboxylate 叔-丁基 4-(氨基甲基)-4-苯基哌啶-1-甲酸基酯 158144-82-2 详细
2-(2-phenoxyphenyl)acetic acid 2-苯氧基苯乙酸 25563-02-4 详细
4-(4-pyridyl)piperidine-4-carbonitrile 4-pyridin-4-ylpiperidine-4-carbonitrile 756452-70-7 详细
3-pyrazin-2-ylphenol 3-(2-吡嗪基)苯酚 570432-61-0 详细
5-[(3S)-5-fluoro-7-hydroxy-3-(isopentylamino)tetralin-6-yl]-1,1-dioxo-1,2,5-thiadiazolidin-3-one 1,2,5-THIADIAZOLIDIN-3-ONE, 5-[(7S)-1-FLUORO-5,6,7,8-TETRAHYDRO-3-HYDROXY-7-[(3-METHYLBUTYL)AMINO]-2 2489404-96-6 详细
tert-butyl 4-fluoro-2-{1H-pyrrolo[2,3-b]pyridin-5-yloxy}benzoate 叔-丁基 4-氟-2-{1H-吡咯并[2,3-b]吡啶-5-氧基}苯酸盐 2007920-25-2 详细
3-[4-(trifluoromethyl)phenoxy]azetidine 3-[4-(三氟甲基)苯氧基]氮杂环丁烷 76263-21-3 详细
4-(4-aminophenoxy)-N-methylpyridine-2-carboxamide 4-(4-氨基苯氧基)-N-甲基-2-吡啶甲酰胺 284462-37-9 详细
1-(4-bromophenyl)cyclopropanesulfonyl chloride 2354862-06-7 详细
2-(2-chloro-4-pyridyl)morpholine;hydrochloride 2940951-05-1 详细
tert-butyl (3S)-3-phenylpiperazine-1-carboxylate 叔-丁基 (3S)-3-苯基哌嗪-1-甲酸基酯 1221274-36-7 详细
1-[3,5-bis(trifluoromethyl)phenyl]-3-[(S)-[(1S,2S,4S,5R)-5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl](6-methoxyquinolin-4-yl)methyl]thiourea 1-[3,5-二(三氟甲基)苯基]-3-[(S)-[(1S,2S,4S,5R)-5-乙烯基-1-氮杂二环[2.2.2]辛烷-2-基](6-甲氧基喹啉-4-基)甲基]硫代脲 852913-16-7 详细
1-[6-(4-fluoropyrazol-1-yl)-3-pyridyl]ethanone 1-[6-(4-fluoro-1H-pyrazol-1-yl)-3-pyridinyl]Ethanone 1980023-94-6 详细
(S)-[(1S,2R,4S,5R)-1-benzyl-5-vinyl-quinuclidin-1-ium-2-yl]-(4-quinolyl)methanol;chloride N-苄基氯化辛可宁 69221-14-3 详细
methyl 2-(rel-(1R,5S,6s)-3-(2-chloro-6-(trifluoromethyl)pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-6-yl)acetate 2-(REL-(1R,5S,6S)-3-(2-氯-6-(三氟甲基)嘧啶-4-基)-3-氮杂双环[3.1.0]己-6-基)乙酸甲酯 2102502-68-9 详细
tert-butyl 3-{[(4-bromophenyl)methyl]amino}piperidine-1-carboxylate 叔-丁基 3-{[(4-溴苯基)甲基]氨基}哌啶-1-甲酸基酯 887584-43-2 详细
1-(6-bromo-5-fluoro-1-methyl-indazol-3-yl)hexahydropyrimidine-2,4-dione 1-(6-溴-5-氟-1-甲基-1H-吲唑-3-基)二氢嘧啶-2,4(1H,3H)-二酮 2760850-50-6 详细
(3R,4R,5R)-3,4-bis[(2,4-dichlorophenyl)methoxy]-5-[(2,4-dichlorophenyl)methoxymethyl]-3-vinyl-tetrahydrofuran-2-one 2940860-88-6 详细
3-[(2S)-morpholin-2-yl]benzoic acid;hydrochloride 2718999-78-9 详细
tripyrrolidin-1-yl(triazolo[4,5-b]pyridin-3-yloxy)phosphonium;hexafluorophosphate (7-氮杂苯并三唑-1-氧)三吡咯磷六氟磷酸盐 156311-83-0 详细
3-(m-tolyl)oxetane-3-carboxylic acid 3-(3-甲基苯基)噁丁环烷-3-羧酸 1393568-32-5 详细
4-chloro-2-{4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,]dodeca-2(6),7-dien-10-yl}pyridine-3-carbaldehyde 1434050-55-1 1434050-55-1 详细
1-pyrimidin-2-ylcyclopropanecarbonitrile 1-(2-pyrimidinyl)cyclopropanecarbonitrile 1378798-49-2 详细
1-(3-methoxyanilino)cyclopropanecarboxylic acid 1 - [(3-甲氧基苯基)氨基]环丙烷-1-羧酸 1252591-26-6 详细
2-(2-methoxyphenyl)pyrimidin-4-yl]methanol 2-(2-甲氧基苯基)嘧啶-4-基]甲醇 1339058-28-4 详细
3-[5-(aminomethyl)-1-oxo-isoindolin-2-yl]piperidine-2,6-dione;hydrochloride 3-(6-氨基亚甲基-3-氧代-1H-异吲哚-2-基)哌啶-2,6-二酮盐酸盐 1158264-69-7 详细
N3-(4-fluorophenyl)pyridine-3,4-diamine N3-(4-氟苯基)吡啶-3,4-二胺 1469018-93-6 详细
tert-butyl 2-(4-methoxycarbonylphenyl)pyrrolidine-1-carboxylate 1-BOC-2-[4-(甲氧基羰基)苯基]吡咯烷 1243198-96-0 详细
6-(2,3-dihydro-1,4-benzodioxin-5-yl)-N-[3-[(dimethylamino)methyl]phenyl]-2-methoxy-pyridin-3-amine 6-(2,3-二氢-1,4-苯并二噁英-5-基)-N-[3-[((二甲氨基)甲基]苯基]-2-甲氧基-吡啶-3-胺 2306268-61-9 详细
1-(1-bicyclo[1.1.1]pentanyl)pyrazole 1-(双环[1.1.1]戊烷-1-基)-1H-吡唑 2417226-01-6 详细
cis-2-phenylcyclopropane-1-carboxylic acid 顺-2-苯基环丙烷-1-羧酸 939-89-9 详细
2-piperazin-1-yl-5-(trifluoromethyl)pyrimidine;hydrochloride 1884156-37-9 详细
4-(4-methylpiperazin-1-yl)sulfonylaniline 4-(4-甲基哌嗪-1-磺酰)苯胺 21623-68-7 详细
1-(2-bromo-4-pyridyl)cyclopropanecarbonitrile 1-(2-BROMOPYRIDIN-4-YL)CYCLOPROPANECARBONITRILE 1279815-46-1 详细
(2R)-2-(2-isopropylphenyl)pyrrolidine (2R)-2-[2-(METHYLETHYL)PHENYL]PYRROLIDINE 1213907-32-4 详细
(4S)-4-phenyl-3-propanoyl-oxazolidin-2-one (S)-4-苯基-3-丙酰基-2-恶唑烷酮 184363-66-4 详细
ethyl 2-[1-[[1-(2-ethoxy-2-oxo-ethyl)cyclopropyl]amino]cyclopropyl]acetate 乙基 2-(1-{[1-(2-乙氧基-2-氧亚基乙基)环丙基]氨基}环丙基)醋酸盐 2007924-94-7 详细
(3R)-N-{3,6-dichloro-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-amine hydrochloride (3R)-N-{3,6-二氯-1H-吡唑并[3,4-d]嘧啶-4-基}哌啶-3-胺盐酸 2007916-10-9 详细
tert-butyl 3-[(4-bromophenyl)methylamino]pyrrolidine-1-carboxylate 叔-丁基 3-{[(4-溴苯基)甲基]氨基}吡咯烷-1-甲酸基酯 1260810-70-5 详细
7-bromo-N-(1,3-dimethylpyrazol-4-yl)quinazolin-2-amine 7-溴-N-(1,3-二甲基吡唑-4-基)喹唑啉-2-胺 2227206-75-7 详细
Diphenylsilane 二苯基硅烷 775-12-2 详细
4-(6-fluoro-2-pyridyl)thiazol-2-amine 4-(6-氟吡啶-2-基)噻唑-2-胺 2422030-89-3 详细
(2R)-2-[(2R)-pyrrolidin-2-yl]pyrrolidine;dihydrochloride 2704188-21-4 详细
2-(1-fluorocyclopropyl)-4-methyl-1H-pyrimidin-6-one 2891599-45-2 详细
2-(4-cyclohexylcyclohex-1-en-1-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 1868137-31-8 详细
3-[5-(2-bromoethoxy)-1-oxo-isoindolin-2-yl]piperidine-2,6-dione 2883559-55-3 详细
(2R)-2-(9H-fluoren-9-ylmethoxycarbonylamino)-3-methyl-3-tritylsulfanyl-butanoic acid Fmoc-S-三苯甲基-L-青霉胺 201531-88-6 详细
1-(3-bromophenyl)cyclopropane-1-carboxylic acid 1-(3-溴苯基)环丙烷-1-羧酸 124276-95-5 详细
tert-butyl 4-(3-amino-1H-pyrazol-5-yl)piperidine-1-carboxylate 叔-丁基 4-(3-氨基-1H-吡唑-5-基)哌啶-1-甲酸基酯 1169563-99-8 详细
(1S)-[1,1'-Binaphthalene]-2,2'-diol S-1,1'-联-2-萘酚 18531-99-2 详细
3-(6-fluoro-3-pyridyl)oxetan-3-amine;hydrochloride 2940945-53-7 详细
5-cyclopropylpyridin-2-amine 5-环丙基吡啶-2-胺 893738-68-6 详细
(3R)-3-(4-bromophenyl)piperidine (R)- 3-(4-溴苯基)哌啶 1336754-69-8 详细
3-(4-methoxyphenyl)oxetan-3-amine;hydrochloride 1332765-59-9 1332765-59-9 详细
trans-2-(6-bromo-3-pyridyl)cyclopropanecarboxylic acid (1S,2S)-rel-2-(6-溴吡啶-3-基)环丙烷-1-羧酸 918305-72-3 详细
5-methyl-1-phenyl-1H-pyrazole-4-sulfonyl chloride 5-甲基-1-苯基-1H-吡唑-4-磺酰氯 342405-38-3 详细
4-(2-aminoethylamino)-2-(2,6-dioxo-3-piperidyl)isoindoline-1,3-dione;2,2,2-trifluoroacetic acid 沙利度胺-NH-C2-NH2三氟醋酸盐 1957235-67-4 详细
2-(2,6-dioxo-3-piperidyl)-5,6-difluoro-isoindoline-1,3-dione 2-(2,6-dioxopiperidin-3-yl)-5,6-difluoroisoindoline-1,3-dione 1496997-41-1 详细
trans-2-[4-(4-ethylcyclohexyl)cyclohexen-1-yl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 1868137-11-4 详细
2-phenyl-1H-imidazole 2-苯基咪唑 670-96-2 详细
tert-butyl 3-cyclopropylpiperazine-1-carboxylate 3-环丙基哌嗪-1-羧酸叔丁酯 886779-85-7 详细
2,4-dichloro-5-cyclopropylpyrimidine 2,4-DICHLORO-5-CYCLOPROPYLPYRIMIDINE 1190379-86-2 详细
n-(tetrahydro-4-phenyl-2h-pyran-4-yl)acetamide n-(四氢-4-苯基-2h-吡喃-4-基)醋胺石 939801-34-0 详细
tert-butyl N-[trans-2-[4-(oxan-2-yloxy)phenyl]cyclopropyl]carbamate 叔-丁基 N-[(1S,2R)-rel-2-[4-(噁烷-2-氧基)苯基]环丙基]氨基甲酯 1946017-76-0 详细
ethyl 1-(3-pyridylmethyl)pyrazole-3-carboxylate ethyl 1-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxylate 2250242-67-0 详细
ethyl 4-(4-pyridyl)-1H-pyrazole-3-carboxylate 1H-Pyrazole-3-carboxylic acid, 4-(4-pyridinyl)-, ethyl ester 1583555-40-1 详细
3-(3-cyano-5-fluoro-phenoxy)-2-(difluoromethyl)-6-methylsulfonyl-benzonitrile Benzonitrile, 3-(3-cyano-5-fluorophenoxy)-2-(difluoromethyl)-6-(methylsulfonyl)- 1672663-84-1 详细
4-[(4-bromophenyl)methyl]morpholine 4-(4-溴苄基)-吗啉 132833-51-3 详细
3-bromo-7-chloro-1-cyclopropyl-4-methyl-1,6-naphthyridin-2-one 2831908-81-5 详细
4,6-dichloro-2-pyrimidin-5-yl-pyrimidine 1858039-72-1 详细
N-(2-chloro-4-nitro-phenyl)-1-hydroxy-naphthalene-2-carboxamide N-(2-氯-4-硝基-苯基)-1-羟基-萘-2-甲酰胺 65570-43-6 详细
tert-butyl N-[cis-2-phenylcyclopropyl]carbamate 叔-丁基 N-[(1R,2R)-rel-2-苯基环丙基]氨基甲酯 847644-86-4 详细
4-[(6-chloro-3-pyridyl)oxy]-6,7-dimethoxy-quinoline 4-((6-氯吡啶-3-基)氧基)-6,7-二甲氧基喹啉 666731-22-2 详细
4-bromo-3-morpholino-benzonitrile 4-bromo-3-morpholinobenzonitrile 2090718-87-7 详细
1-pyrrolidin-2-ylcyclopropanol hydrochloride 1-pyrrolidin-2-ylcyclopropanol hydrochloride 2191401-19-9 详细
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