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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
(2R,3R,4R,5R)-3,4-dibenzoyloxy-5-(5-methyl-4-oxo-2-thioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methyl benzoate O2',O3',O5'-三苯甲酰基-5-甲基-2-硫代尿苷 75921-08-3 详细
methyl 2-[(1R)-1-phenylethyl]-2-azabicyclo[2.2.1]hept-5-ene-3-carboxylate 详细
trans-4-(3-amino-2,2,4,4-tetramethyl-cyclobutoxy)benzonitrile;hydrochloride 2940879-73-0 详细
1-benzyl-4-phenyl-3,6-dihydro-2H-pyridine 1-苄基-4-苯基-1,2,3,6-四氢吡啶 38025-45-5 详细
3-cyclopropylazetidin-3-ol hydrochloride 3-环丙基吖丁啶-3-醇盐酸 848192-93-8 详细
3-Boc-amino-3-(4-bromophenyl)oxetane tert-Butyl (3-(4-bromophenyl)oxetan-3-yl)carbamate 1279090-24-2 详细
3-(4-methoxyphenyl)oxetane-3-carboxylic acid 3-(4-甲氧苯基)噁丁环烷-3-羧酸 1416323-25-5 详细
(5-cyclopropylpyridin-2-yl)methanol (5-环丙基吡啶-2-基)甲醇 1301168-21-7 详细
4-(pyridin-3-yloxy)benzoic acid 4-(吡啶-3-基氧基)苯甲酸 437383-99-8 详细
1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)cyclopropane-1-carboxylic acid 1-(2,2-二氟苯并[D][1,3]二氧杂环戊烯-5-基)环丙烷甲酸 862574-88-7 详细
methyl 3-cyclopropyl-1H-pyrazole-4-carboxylate METHYL 5-CYCLOPROPYLPYRAZOLE-4-CARBOXYLATE 1150164-05-8 详细
2-methyl-5-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-1,3,4-oxadiazole 2-甲基-5-[4-(四甲基-1,3,2-二噁硼戊环-2-基)苯基]-1,3,4-噁二唑 1056456-24-6 详细
N-(oxetan-3-yl)oxetan-3-amine N-(噁丁环烷-3-基)噁丁环烷-3-胺 1057682-66-2 详细
3-(3-bromophenyl)oxetane 3-(3-溴苯基)噁丁环烷 1044507-52-9 详细
5-bromo-7-[trans-4-(tert-butyldimethylsilanyloxy)cyclohexyl]-2-chloro-7h-pyrrolo[2,3-d]pyrimidine 5-溴-7-[反-4-(叔-丁基二甲基硅烷氧基)环己基]-2-氯-7h-吡咯并[2,3-d]嘧啶 1392804-15-7 详细
3-(4-fluorophenyl)oxetan-3-amine hydrochloride 3-(4-氟苯基)噁丁环烷-3-胺盐酸 1332839-79-8 详细
1-(pyrimidin-2-yl)cyclopropan-1-amine dihydrochloride 1-(嘧啶-2-基)环丙烷-1-胺二盐酸 1159734-42-5 详细
(3S)-3-phenylpyrrolidine hydrochloride (S)-3-苯基吡咯烷盐酸盐 1094670-20-8 详细
5-(2-chlorophenyl)cyclohexane-1,3-dione 5-(2-氯苯基)环己烷-1,3-二酮 55579-68-5 详细
1-{6-bromopyrazolo[1,5-a]pyridin-3-yl}-1,3-diazinane-2,4-dione 2925080-89-1 详细
4-(4-methoxyphenyl)-2-oxabicyclo[2.1.1]hexane-5-carboxylic acid 2171880-95-6 详细
tert-butyl 4-(3-ethynylazetidine-1-carbonyl)-3,3-difluoropiperidine-1-carboxylate 详细
1-tert-butoxycarbonyl-4-cyclopropyl-piperidine-4-carboxylic acid 1-[(叔-丁氧基)羰基]-4-环丙基哌啶-4-羧酸 1346599-08-3 详细
2-phenyl-2,6-diazaspiro[3.3]heptan-1-one 2-苯基-2,6-二氮杂螺[3.3]庚烷-1-酮 960079-47-4 详细
tert-butyl 3-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]azetidine-1-carboxylate 3-[4-(四甲基-1,3,2-二氧杂硼烷-2-基)-1H-吡唑-1-基]氮杂环丁烷-1-羧酸叔丁酯 877399-35-4 详细
1-pyrimidin-2-ylazetidin-3-amine;dihydrochloride 1-(嘧啶-2-基)吖丁啶-3-胺二盐酸 1365968-57-5 详细
methyl (1S,3S,4R)-2-[(1R)-1-phenylethyl]-2-azabicyclo[2.2.1]hept-5-ene-3-carboxylate (1S,3S,4R)-2-((1R)-1-苯基乙基)-2-氮杂双环[2.2.1]庚-5-烯-3-羧酸甲酯 130194-96-6 详细
methyl 1-(pyrazin-2-yl)cyclopropane-1-carboxylate 甲基 1-(吡嗪-2-基)环丙烷-1-甲酸基酯 1363382-27-7 详细
2-Aminoadenosine 2-氨基腺嘌呤核苷 2096-10-8 详细
N'-(2-methylnaphthalen-1-yl)-N-[(pyridin-2-yl)methyl]ethanediamide N1-(2-吡啶甲基)-N2-(2-甲基-1-萘基)草酰胺 2611225-93-3 详细
(1S)-1-[6-(4-fluoropyrazol-1-yl)-3-pyridyl]ethanamine;hydrochloride (S)-1-(6-(4-氟-1H-吡唑-1-基)吡啶-3-基)乙-1-胺盐酸盐 2097133-17-8 详细
5′-O-[Bis(4-methoxyphenyl)phenylmethyl]-2′-O-methyl-N-(2-methyl-1-oxopropyl)guanosine 5'-O-DMT-N2-异丁酰基-2'-O-甲基鸟苷 114745-26-5 详细
methyl (1S,3R)-2-(2-chloroacetyl)-1-(4-methylsulfonylphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-3-carboxylate 化合物 GPX4-IN-4 2920221-53-8 详细
tert-butyl 3-[4-(trifluoromethyl)phenyl]piperazine-1-carboxylate 叔-丁基 3-[4-(三氟甲基)苯基]哌嗪-1-甲酸基酯 886767-93-7 详细
tert-butyl 4-(1-methoxycyclopropanecarbonyl)piperazine-1-carboxylate 叔-丁基 4-(1-甲氧基环丙羰基)哌嗪-1-甲酸基酯 1788041-47-3 详细
2'-Deoxyuridine 2-脱氧尿苷 951-78-0 详细
1-(4-bromophenyl)pyrimidine-2,4-dione 53727-25-6 详细
3-phenoxyazetidine hydrochloride 3-苯氧基吖啶盐酸盐 301335-39-7 详细
4-chloro-6-phenylpyrimidin-2-amine 2-氨基-4-氯-6-苯基嘧啶 36314-97-3 详细
N'-[9-[(2R,4S,5R)-5-[[bis(4-methoxyphenyl)-phenyl-methoxy]methyl]-4-[2-cyanoethoxy-(diisopropylamino)phosphanyl]oxy-tetrahydrofuran-2-yl]-6-oxo-3H-purin-2-yl]-N,N-dimethyl-formamidine DMF-DG-CE亚磷酰胺单体 330628-04-1 详细
tert-butyl 4-(4-amino-3-methoxy-phenyl)piperazine-1-carboxylate 4-(4-氨基-3-甲氧基苯基)哌嗪-1-羧酸叔丁酯 1246532-96-6 详细
bis(adamantan-1-yl)(2-{[tris(propan-2-yl)silyl]oxy}phenyl)phosphane DI(1-ADAMANTYL)-(2-TRIISOPROPYLSILOXYPHENYL)PHOSPHINE 1384966-55-5 详细
4-bromo-1-(oxetan-3-yl)-1,2-dihydropyridin-2-one 4-溴-1-(氧杂环丁烷-3-基)吡啶-2(1H)-酮 1352754-13-2 详细
tert-butyl 4-(4-aminophenyl)piperidine-1-carboxylate 1-BOC-4-(4-氨基苯基)哌啶 170011-57-1 详细
tert-butyl 3-(4-piperidyl)azetidine-1-carboxylate;hydrochloride 2752183-78-9 详细
tert-butyl N-(1-pyrazin-2-ylcyclopropyl)carbamate 2809035-71-8 详细
2-(3-methylazetidin-3-yl)pyridine 2,2,2-trifluoroacetic acid 2940961-42-0 详细
4-(1H-1,2,3,4-tetrazol-1-yl)phenol 4-(1H-1,2,3,4-四唑-1-基)苯酚 64001-11-2 详细
1-((4-Fluorophenyl)carbamoyl)cyclopropanecarboxylic acid 1-(4-氟苯基氨基甲酰基)环丙烷羧酸 849217-48-7 详细
ethyl 3-cyclopropyl-1H-pyrazole-4-carboxylate 乙基 3-环丙基-1H-吡唑-4-甲酸基酯 1246471-38-4 详细
1-(5-fluoropyridin-2-yl)cyclopropane-1-carboxylic acid 1302580-98-8 1302580-98-8 详细
(2R)-2-(2-methoxyphenyl)-2-(oxan-4-yloxy)ethan-1-ol (2R)-2-(2-甲氧苯基)-2-(噁烷-4-氧基)乙烷-1-醇 1434652-66-0 详细
3-[[(2R,3R,4R,5R)-2-[[bis(4-methoxyphenyl)-phenyl-methoxy]methyl]-5-(2,4-dioxopyrimidin-1-yl)-4-methoxy-tetrahydrofuran-3-yl]oxy-(diisopropylamino)phosphanyl]oxypropanenitrile 2’-OMe-U亚磷酰胺单体 110764-79-9 详细
4-(4,6-dimethoxy-1,3,5-triazin-2-yl)-4-methyl-morpholin-4-ium;chloride 4-(4,6-二甲氧基三嗪-2-基)-4-甲基吗啉盐酸盐 3945-69-5 详细
1-(3-methylazetidin-3-yl)piperidine;dihydrochloride 2322925-08-4 详细
N-[9-[(2R,4S,5R)-5-[[bis(4-methoxyphenyl)-phenyl-methoxy]methyl]-4-[2-cyanoethoxy-(diisopropylamino)phosphanyl]oxy-tetrahydrofuran-2-yl]purin-6-yl]benzamide 5'-O-(4,4'-二甲氧基三苯基)-N6-苯甲酰基-2'-脱氧腺苷-3'-(2-氰乙基-N,N-二异丙基)亚磷酰胺 98796-53-3 详细
1-[(2S,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-5-methyl-2-thioxo-pyrimidin-4-one 2940859-47-0 详细
methyl 1-(3-chloro-4-pyridyl)-3-oxo-cyclobutanecarboxylate 详细
3-(4-bromophenyl)oxetan-3-ol 3-(4-溴苯基)噁丁环烷-3-醇 1093878-32-0 详细
tert-butyl 3-(1-aminocyclopropyl)azetidine-1-carboxylate 叔-丁基 3-(1-氨基环丙基)吖丁啶-1-甲酸基酯 1352012-69-1 详细
tert-butyl 3-(4-hydroxy-1-piperidyl)azetidine-1-carboxylate 178311-46-1 详细
3-phenylcyclobutan-1-amine 3-苯基环丁烷-1-胺 90874-41-2 详细
3-methyl-4-{[1,2,4]triazolo[1,5-a]pyridin-7-yloxy}aniline 4-([1,2,4]三唑[1,5-A]吡啶-7-氧基)-3-甲基苯胺 937263-71-3 详细
4-(anthracen-9-yl)-3-tert-butyl-2,3-dihydro-1,3-benzoxaphosphole 4-(9-蒽基)-3-(叔丁基)-2,3-二氢苯并[D][1,3]氧,膦戊轭 1268693-24-8 详细
1-(pyrimidin-5-yl)azetidin-3-amine hydrochloride 1-(嘧啶-5-基)吖丁啶-3-胺盐酸 2173991-64-3 详细
3-(5-bromo-6-fluoro-1-oxo-isoindolin-2-yl)piperidine-2,6-dione 3-(5-溴-6-氟-1-氧异喹啉-2-基)哌啶-2,6-二酮 2409005-96-3 详细
2-[4-(2,6-dioxo-3-piperidyl)phenoxy]acetic acid 2-(4-(2,6-二氧代哌啶-3-基)苯氧基)乙酸 2782024-58-0 详细
Inosine 肌苷 58-63-9 详细
1-phenylazetidin-3-ol 1-苯偶氮基丁啶-3-醇 857280-53-6 详细
4-(oxetan-3-yloxy)aniline 4-(噁丁环烷-3-氧基)苯胺 1349715-80-5 详细
3-(5-hydroxy-1-oxo-isoindolin-2-yl)piperidine-2,6-dione 3-(5-羟基-1-氧代异吲哚-2-基)哌啶-2,6-二酮 1416990-08-3 详细
3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine-7-carbaldehyde 3-(CYCLOPROPYLMETHYL)-8-(TRIFLUOROMETHYL)-[1,2,4]TRIAZOLO[4,3-A]PYRIDINE-7-CARBALDEHYDE 1254982-03-0 详细
5-bromo-2,2'-bipyridine 5-溴-2,2'-联吡啶 15862-19-8 详细
(5R)-5-benzyl-2,2,3-trimethyl-imidazolidin-4-one hydrochloride (5R)-(+)-2,2,3-三甲基-5-苄基-4-咪唑啉酮单盐酸盐 323196-43-6 详细
2-amino-8-bromo-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-6,9-dihydro-3H-purin-6-one 8-溴鸟苷 4016-63-1 详细
hemi(oxalic acid);3-(oxetan-3-yl)pyrrolidine 2940956-82-9 详细
3-cyclobutyl-1H-pyrazol-5-amine 3-环丁基-1H-吡唑-5-胺 326827-21-8 详细
5-phenylthiazole 5-苯基噻唑 1826-13-7 详细
methyl (3S)-5-oxo-1-[(1R)-1-phenylethyl]pyrrolidine-3-carboxylate 甲基 (3s)-5-氧亚基-1-[(1r)-1-苯基乙基]吡咯烷-3-甲酸基酯 99735-46-3 详细
N-Benzoyl-5′-O-[bis(4-methoxyphenyl)phenylmethyl]-2′-deoxyadenosine N6-苯甲酰基-5'-O-(4,4'-二甲氧基三苯基)-2'-脱氧腺苷 64325-78-6 详细
(NE)-N-(piperidine-1-carbonylimino)piperidine-1-carboxamide (NE)-N-{[(E)-哌啶-1-羰基]氨亚基}哌啶-1-甲酰胺 10465-81-3 详细
3-cyclopropyl-1H-pyrazol-5-amine 3-环丙基-1H-吡唑-5-胺 175137-46-9 详细
N-{1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-2-oxo-1,2-dihydropyrimidin-4-yl}benzamide 苯甲酰胞苷 13089-48-0 详细
1-cyclobutylpiperazine dihydrochloride 二盐酸1-环丁基哌嗪 799557-65-6 详细
3-cyclopropylbicyclo[1.1.1]pentan-1-amine;hydrochloride 2763756-42-7 详细
methyl 3-cyclopropylbicyclo[1.1.1]pentane-1-carboxylate 2940939-17-1 详细
tert-butyl 4-[(5-bromo-2-chloro-4-pyridyl)methyl]-4-hydroxy-piperidine-1-carboxylate 2771352-36-2 详细
tert-butyl (2R,5S)-2-(1,3-benzothiazol-5-yl)-5-methyl-piperidine-1-carboxylate 2760268-03-7 详细
N-[1-[(2R,4S,5R)-5-[[bis(4-methoxyphenyl)-phenyl-methoxy]methyl]-4-[2-cyanoethoxy-(diisopropylamino)phosphanyl]oxy-tetrahydrofuran-2-yl]-2-oxo-pyrimidin-4-yl]benzamide DMT-dC(bz)亚磷酰胺单体 102212-98-6 详细
tofacitinib citrate 枸橼酸托法替尼 540737-29-9 详细
tert-butyl N-[1-(4-bromophenyl)cyclopropyl]carbamate 1-(4-溴苯基)-环丙基]氨基甲酸叔丁酯 360773-84-8 详细
tert-butyl (4S)-2,2-dioxo-4-phenyl-1,2λ,3-oxathiazolidine-3-carboxylate 叔-丁基 (4S)-2,2-二氧亚基-4-苯基-1,2λ?,3-氧杂噻唑烷-3-甲酸基酯 479687-23-5 详细
(3R)-3-(benzenesulfonyl)pyrrolidine (3R)-3-(苯磺酰)吡咯烷 1268521-39-6 详细
3-(3-fluorophenyl)oxetane-3-carboxylic acid 3-(3-Fluorophenyl)oxetane-3-carboxylic acid 1393553-52-0 详细
N-[1-[(2R,4S,5R)-5-[[bis(4-methoxyphenyl)-phenyl-methoxy]methyl]-4-[2-cyanoethoxy-(diisopropylamino)phosphanyl]oxy-tetrahydrofuran-2-yl]-5-methyl-2-oxo-pyrimidin-4-yl]benzamide Bz-5-ME-2'-脱氧胞苷亚磷酰胺单体 105931-57-5 详细
1-(5-bromopyridin-3-yl)cyclopropan-1-amine hydrochloride 1-(5-溴吡啶-3-基)环丙烷-1-胺盐酸 1993189-05-1 详细
3-[[(2R,3S,5R)-2-[[bis(4-methoxyphenyl)-phenyl-methoxy]methyl]-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-3-yl]oxy-(diisopropylamino)phosphanyl]oxypropanenitrile 5'-(4,4'-二甲氧基三苯基)-3'-脱氧胸苷 2'-(2-氰乙基-N,N-二异丙基)亚磷酰胺 98796-51-1 详细
(3S)-N-(oxetan-3-yl)pyrrolidin-3-amine dihydrochloride (3S)-N-(噁丁环烷-3-基)吡咯烷-3-胺二盐酸 2173637-22-2 详细
5′-O-(4,4′-Dimethoxytrityl)thymidine 保护胸苷 40615-39-2 详细
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