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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
1-(pyrazin-2-yl)cyclopropane-1-carboxylic acid 1-(吡嗪-2-基)环丙烷-1-羧酸 1159734-52-7 详细
1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)cyclopropane-1-carbonitrile 1-(2,2-二氟-2H-1,3-苯并二噁戊环-5-基)环丙烷-1-甲腈 862574-87-6 详细
3-nitro-4-[(oxan-4-ylmethyl)amino]benzene-1-sulfonamide 3-硝基-4-[(噁烷-4-基甲基)氨基]苯-1-磺酰胺 1228779-96-1 详细
(3S)-3-(benzenesulfonyl)pyrrolidine (3S)-3-(苯磺酰)吡咯烷 1408057-40-8 详细
tert-butyl 4-(1-hydroxycyclopropanecarbonyl)piperazine-1-carboxylate 叔-丁基 4-(1-羟基环丙羰基)哌嗪-1-甲酸基酯 1788054-84-1 详细
benzyl N-[1-(5-chloropyrimidin-2-yl)cyclopropyl]carbamate (1-(5-氯嘧啶-2-基)环丙基)氨基甲酸苄酯 1422356-97-5 详细
4-bromo-1-cyclopropylpyridin-2(1H)-one 4-溴-1-环丙基吡啶-2(1H)-酮 1193334-86-9 详细
N-[9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]purin-6-yl]benzamide N6-苯甲酰基腺苷 4546-55-8 详细
tert-butyl 3-hydroxy-3-[(pyridin-2-yl)methyl]azetidine-1-carboxylate 3-羟基-3-[(吡啶-2-基)甲基]氮杂环丁烷-1-羧酸叔丁酯 1490206-48-8 详细
tert-butyl 4-(azetidin-3-yloxy)piperidine-1-carboxylate hydrochloride 2306278-50-0 详细
3-(6-bromo-1-methyl-1H-indazol-3-yl)piperidine-2,6-dione 3-(6-溴-1-甲基-1H-吲唑-3-基)哌啶-2,6-二酮 2913408-82-7 详细
1-(4-aminophenyl)piperidin-4-ol 1-(4-氨基苯基)-4-羟基哌啶 142752-12-3 详细
tert-butyl (2S)-2-(4-bromo-1H-imidazol-2-yl)pyrrolidine-1-carboxylate 叔-丁基 (2S)-2-(4-溴-1H-咪唑-2-基)吡咯烷-1-甲酸基酯 1007882-59-8 详细
2-chloro-3-(1,3-dithian-2-yl)pyrazine 2-氯-3-(1,3-二硫烷-2-基)吡嗪 874114-28-0 详细
5-(azetidin-3-yl)-2H-1,2,3,4-tetrazole hydrochloride 5-(吖丁啶-3-基)-2H-1,2,3,4-四唑盐酸 950691-49-3 详细
(2R)-2-methyl-1-[(1S)-1-phenylethyl]piperidin-4-one (2R)-2-甲基-1-[(1S)-1-苯基乙基]哌啶-4-酮 89467-37-8 详细
1-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazine dihydrochloride 1 - {[2-(4-氯苯基)-4,4-二甲基环己-1-烯-1-基]甲基}哌嗪二盐酸盐 1628047-87-9 详细
4-(cyclohex-1-en-1-yl)-3-(trifluoromethyl)benzoic acid 4-(环己三烯-1-烯-1-基)-3-(三氟甲基)苯甲酸 1034188-31-2 详细
3-phenylbicyclo[1.1.1]pentan-1-amine hydrochloride 3-Phenylbicyclo[1.1.1]pentan-1-aminehydrochloride 83249-11-0 详细
2-chloro-5-[(1-methylpiperidin-4-yl)methoxy]pyrimidine 2-氯-5-[(1-甲基哌啶-4-基)甲氧基]嘧啶 1408074-71-4 详细
3-phenylpiperidine-3-carboxylic acid 116140-39-7 详细
3-(2-fluorophenyl)oxetan-3-yl]methanamine [3-(2-FLUOROPHENYL)OXETAN-3-YL]METHANAMINE 1507868-26-9 详细
1-β-D-Arabinofuranosyl-5-methyl-2,4(1H,3H)-pyrimidinedione 阿糖胸苷 605-23-2 详细
5-amino-1-(oxan-4-yl)-1H-pyrazole-4-carboxamide 5-氨基-1-(噁烷-4-基)-1H-吡唑-4-甲酰胺 1082745-50-3 详细
methyl 3-(4-chlorophenyl)pyrazine-2-carboxylate 甲基 3-(4-氯苯基)吡嗪-2-甲酸基酯 1363382-34-6 详细
5-methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acid 5-甲基-2-(2H-1,2,3-三唑-2-基)苯甲酸 956317-36-5 详细
(3S)-1-{[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methyl}pyrrolidin-3-ol (S)-1-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)pyrrolidin-3-ol 1206641-40-8 详细
(6aR,8R,9R,9aS)-8-(6-aminopurin-9-yl)-2,2,4,4-tetraisopropyl-6a,8,9,9a-tetrahydro-6H-furo[3,2-f][1,3,5,2,4]trioxadisilocin-9-ol 3,5-O-(1,1,3,3-四异丙基-1,3-二硅氧烷)腺苷 69304-45-6 详细
3-(7-bromo-1-oxo-isoindolin-2-yl)piperidine-2,6-dione 3-(7-溴-1-氧亚基-2,3-二氢-1H-异吲哚-2-基)哌啶-2,6-二酮 2229976-08-1 详细
tert-butyl 3-(2-fluoro-5-methylphenyl)-3-hydroxyazetidine-1-carboxylate 3-(2-氟-5-甲基苯基)-3-羟基氮杂环丁烷-1-羧酸叔丁酯 1493550-86-9 详细
methyl 4-(4-methoxyphenyl)-2-oxabicyclo[2.1.1]hexane-5-carboxylate 2763776-92-5 详细
1-phenyl-1,6-diazaspiro[3.3]heptane 1-苯基-1,6-二氮杂螺[3.3]庚烷 1363383-39-4 详细
tert-butyl N-[3-(4-cyanophenyl)oxetan-3-yl]carbamate 叔-丁基 N-[3-(4-氰基苯基)噁丁环烷-3-基]氨基甲酯 1158098-77-1 详细
5-(azetidin-3-yl)-2H-1,2,3,4-tetrazole 5-(吖丁啶-3-基)-2H-1,2,3,4-四唑 950725-13-0 详细
5,7-dichloro-2-cyclopropyl-2H-pyrazolo[4,3-d]pyrimidine 5,7-二氯-2-环丙基-2H-吡唑并[4,3-d]嘧啶 1630906-84-1 详细
tert-butyl N-{9-[(3aR,4R,6R,6aR)-6-(hydroxymethyl)-2,2-dimethyl-tetrahydro-2H-furo[3,4-d][1,3]dioxol-4-yl]-9H-purin-6-yl}-N-[(tert-butoxy)carbonyl]carbamate 叔-丁基 N-{9-[(3aR,4R,6R,6aR)-6-(羟甲基)-2,2-二甲基-四氢-2H-呋喃并[3,4-d][1,3]二噁戊环-4-基]-9H-嘌呤-6-基}-N-[(叔-丁氧基)羰基]氨基甲酯 1152172-19-4 详细
4-(oxetan-3-yl)piperidine hemioxalate 4-(噁丁环烷-3-基)哌啶半草酸酯 1523606-46-3 详细
3-[(1S)-1-aminoethyl]-8-chloro-2-phenyl-1,2-dihydroisoquinolin-1-one 3-[(1S)-1-氨基乙基]-8-氯-2-苯基-1,2-二氢异喹啉-1-酮 1350643-72-9 详细
2-chloro-4-(1H-pyrazol-3-yl)benzonitrile 2-氯-4-(1H-吡唑-3-基)苯甲腈 1297537-37-1 详细
(7S)-7-(pyrrolidin-1-yl)-6,7,8,9-tetrahydro-5H-benzo[7]annulen-2-amine CPD3615-A5 2045894-03-7 详细
4-(azetidine-3-carbonyl)morpholine hydrochloride 4-(吖丁啶-3-羰基)吗啉盐酸 1619991-15-9 详细
1-(azetidine-3-carbonyl)piperidin-4-ol hydrochloride 1-(吖丁啶-3-羰基)哌啶-4-醇盐酸 2227204-99-9 详细
1-(3,5-dimethoxyphenyl)piperazine hydrochloride 1-(3,5-DIMETHOXYPHENYL)PIPERAZINE hydrochloride 1993148-46-1 详细
6-[(6-methoxy-3-pyridyl)methyl]-3,6-diazabicyclo[3.1.1]heptane 6-[(6-甲氧基-3-吡啶基)甲基]-3,6-二氮杂双环[3.1.1]庚烷 2306275-33-0 详细
2-(oxetan-3-yloxy)pyrimidin-5-amine 2-(噁丁环烷-3-氧基)嘧啶-5-胺 1349709-06-3 详细
3-(3-methylphenyl)oxetan-3-yl]methanol 3-(3-甲基苯基)噁丁环烷-3-基]甲醇 1904269-10-8 详细
4-(4-chloro-6-methoxy-9H-pyrimido[4,5-b]indol-7-yl)-3,5-dimethyl-isoxazole 4-(4-氯-6-甲氧基-9H-嘧啶基[4,5-B]吲哚-7-基)-3,5-二甲基-异噁唑 1627721-56-5 详细
4-(tetrazol-5-yl)phenylboronic acid 4-(四唑-5-基)苯基硼酸 179942-55-3 详细
N-methyl-N-[(3R,4R)-4-methyl-3-piperidyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine;dihydrochloride N-甲基-N-((3R,4R)-4-甲基哌啶-3-基)-7H-吡咯并[2,3-D]嘧啶-4-胺二盐酸盐 1655430-59-3 详细
tert-butyl 3-(5-bromo-2-pyridyl)-3,6-diazabicyclo[3.1.1]heptane-6-carboxylate 3-(5-溴吡啶-2-基)-3,6-二氮杂双环[3.1.1]庚烷-6-羧酸叔丁酯 2222757-10-8 详细
3-phenylbicyclo[1.1.1]pentane-1-carboxylic acid 3-苯基二环[1.1.1]戊烷-1-羧酸 83249-04-1 详细
3-phenylcyclobutan-1-one 3-苯基环丁烷-1-酮 52784-31-3 详细
(2S,5R)-5-(6-amino-9H-purin-9-yl)-2,5-dihydrofuran-2-yl]methanol (2S,5R)-5-(6-氨基-9H-嘌呤-9-基)-2,5-二氢呋喃-2-基]甲醇 7057-48-9 详细
2,5-dichloro-N-[2-(propane-2-sulfonyl)phenyl]pyrimidin-4-amine 2,5-二氯-N-[2-[(1-甲基乙基)磺酰基]苯基]-4-嘧啶胺 761440-16-8 详细
4-(2H-1,2,3,4-tetrazol-5-yl)piperidine 4-(2H-1,2,3,4-四唑-5-基)哌啶 112626-97-8 详细
ethyl 5-methyl-4-phenoxypyrrolo[2,1-f][1,2,4]triazine-6-carboxylate 乙基 5-甲基-4-苯氧基吡咯并[2,1-f][1,2,4]三嗪-6-甲酸基酯 1363380-63-5 详细
1-(pyrimidin-2-yl)cyclopropan-1-amine 1-(嘧啶-2-基)环丙烷-1-胺 1159878-06-4 详细
5-(2-fluorophenyl)-1H-pyrrole-3-carbaldehyde 5-(2-氟苯基)-1H-吡咯-3-甲醛 881674-56-2 详细
1-(4-bromo-3-fluorophenyl)cyclopropane-1-carbonitrile 1-(4-溴-3-氟苯基)环丙烷甲腈 749269-73-6 详细
3-(4-hydroxy-1-oxo-isoindolin-2-yl)piperidine-2,6-dione 3-(4-hydroxy-1-oxo-1,3-dihydroisoindol-2-yl)piperidine-2,6-dione 1061604-41-8 详细
3-hydroxy-3-[(2S)-2-piperidyl]azetidin-1-yl]-(2,3,4-trifluorophenyl)methanone;hydrochloride 3-羟基-3-[(2S)-2-哌啶基]氮杂环丁烷-1-基]-(2,3,4-三氟苯基)甲酮盐酸盐 2065147-70-6 详细
8-fluoro-1-methyl-3-[2-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]quinazoline-2,4-dione 8-fluoro-1-methyl-3-[2-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]quinazoline-2,4-dione 1643136-29-1 详细
tert-butyl 4-(5-nitropyridin-2-yl)piperazine-1-carboxylate 叔-丁基 4-(5-硝基吡啶-2-基)哌嗪-1-甲酸基酯 193902-78-2 详细
4-[2-[2-[2-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxo-3-piperidyl)isoindoline-1,3-dione 4-((20-叠氮基-3,6,9,12,15,18-六氧杂二十烷基)氨基)-2-(2,6-二氧代哌啶-3-基)异吲哚啉-1,3-二酮 2624181-62-8 详细
3-(azetidin-3-yl)-2-methyl-pyridine dihydrochloride 2937994-79-9 详细
tert-butyl (2S)-2-(1H-imidazol-2-yl)pyrrolidine-1-carboxylate 叔-丁基 (2S)-2-(1H-咪唑-2-基)吡咯烷-1-甲酸基酯 1007882-58-7 详细
3-(oxetan-3-yl)pyrrolidine 3-(噁丁环烷-3-基)吡咯烷 1273567-00-2 详细
6-cyclopropyl-8-fluoro-1,2-dihydroisoquinolin-1-one 6-环丙基-8-氟-1,2-二氢异喹啉-1-酮 1242156-53-1 详细
3-(4-fluorophenyl)-2,4-dioxo-1-(propan-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid 3-(4-FLUOROPHENYL)-1-ISOPROPYL-2,4-DIOXO-1,2,3,4-TETRAHYDROPYRIMIDINE- 5-CARBOXYLIC ACID 1437323-26-6 详细
3-(1-tert-butoxycarbonyl-4-piperidyl)benzoic acid 1-BOC-4-(3-羧基苯基)哌啶 828243-30-7 详细
2-[3-[(tert-butoxycarbonylamino)methyl]phenyl]-5-(trifluoromethyl)pyrazole-3-carboxylic acid 1-[3-[[[(1,1-DIMETHYLETHOXY)CARBONYL]AMINO]METHYL]PHENYL]-3-(TRIFLUOROMETHYL)-1H-PYRAZOLE-5-CARBOXYLIC ACID 640287-99-6 详细
2-[(4-fluorophenyl)methyl]thiophene 2-[(4-氟苯基)甲基]噻吩 63877-96-3 详细
6-[(4-fluorophenyl)methyl]-3,3-dimethyl-1,2-dihydropyrrolo[3,2-b]pyridin-5-yl]methanol 6-[(4-氟苯基)甲基] -3,3-二甲基-1,2-二氢吡咯并[3,2-B]吡啶-5-基]甲醇 1799327-42-6 详细
3-(2-fluoro-5-methyl-phenyl)azetidin-3-ol;hydrochloride hydrochloride 2387602-61-9 详细
(2S)-2-phenylpyrrolidine (S)-2-苯基吡咯烷 59347-91-0 详细
1-pyrazin-2-ylcyclopropanamine;dihydrochloride 2802785-15-3 详细
4-bromo-2-(cyclopropoxy)pyridine 4-溴-2-环丙氧基吡啶 1209460-14-9 详细
4-(oxetan-3-yloxy)phenyl]methanamine 4-(噁丁环烷-3-氧基)苯基]甲胺 1349719-23-8 详细
2-[[(2S)-oxiran-2-yl]methyl]isoindoline-1,3-dione (S)-N-缩水甘油邻苯二甲酰亚胺 161596-47-0 详细
3-(4-bromophenyl)-1-methyl-1,2,4-triazole 3-(4-溴苯基)-1-甲基-1H-1,2,4-三唑 1184174-04-6 详细
(2S)-2-[4-(trifluoromethyl)phenyl]morpholine (2S)-2-[4-(三氟甲基)苯基]吗啉 2349772-26-3 详细
5-bromo-3-cyclopropyl-1H-indazole 5-溴-3-环丙基-1H-吲唑 911305-80-1 详细
5-(3,3-difluorocyclobutyl)-1H-pyrazol-3-amine 5-(3,3-二氟环丁基)-1H-吡唑-3-胺 1425931-95-8 详细
3-cyclopentyl-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]propanenitrile 3-环戊基-3-[4-(4,4,5,5-四甲基-1,3,2-二噁硼戊环-2-基)-1H-吡唑-1-基]丙腈 1153949-38-2 详细
4-[(4-bromo-3-fluorophenyl)methyl]-1λ-thiomorpholine-1,1-dione 4-[(4-溴-3-氟苯基)甲基]-1λ?-硫代吗啉-1,1-二酮 1973485-27-6 详细
tert-butyl 3-[4-fluoro-3-(trifluoromethyl)phenyl]-3-hydroxyazetidine-1-carboxylate 3-[4-氟-3-(三氟甲基)苯基]-3-羟基氮杂环丁烷-1-羧酸叔丁酯 1694286-57-1 详细
1-(3,5-difluorobenzoyl)piperazine hydrochloride 1-(3,5-二氟苯甲酰)哌嗪盐酸 1580741-84-9 详细
3-(4-bromophenyl)piperidine-2,6-dione 3-(4-溴苯基)哌啶-2,6-二酮 1267337-47-2 详细
9-bromo-7-methyl-2-(morpholin-4-yl)-4H-pyrido[1,2-a]pyrimidin-4-one 9-溴-7-甲基-2-(吗啉-4-基)-4H-吡啶并[1,2-a]嘧啶-4-酮 351002-16-9 详细
4-(oxan-4-yl)aniline 4-(四氢吡喃-4-基)苯胺 62071-40-3 详细
ethyl 2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]acetate 乙基 2-[4-(吗啉-4-基)-6-氧亚基-1,6-二氢嘧啶-2-基]醋酸盐 1260543-99-4 详细
trans-2-(5-bromo-2-thienyl)cyclopropanecarboxylic acid (1S,2S)-rel-2-(5-溴噻吩-2-基)环丙烷-1-羧酸 1818257-71-4 详细
5-[trans-2-aminocyclopropyl]thiophene-2-carboxylic acid;hydrochloride 5-[(1S,2S)-rel-2-氨基环丙基]噻吩-2-羧酸盐酸 2055841-95-5 详细
4-bromo-2-(2,6-dioxo-3-piperidyl)isoindoline-1,3-dione 4-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione 2093536-12-8 详细
1-(3-bromophenyl)cyclopropane-1-carbonitrile 1-(3-溴苯基)环丙烷-1-甲腈 124276-83-1 详细
4-(2,4-dioxohexahydropyrimidin-1-yl)benzoic acid 4-(2,4-二氧亚基六氢嘧啶-1-基)苯甲酸 2599846-40-7 详细
3-[4-(trifluoromethyl)phenyl]azetidin-3-ol;hydrochloride 3-[4-(三氟甲基)苯基]-3-氮杂环丁烷醇盐酸盐 2751620-36-5 详细
4-{[5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazol-4-yl]methoxy}piperidine 4-{[5-环丙基-3-(2,6-二氯苯基)-1,2-噁唑-4-基]甲氧基}哌啶 1103501-11-6 详细
3-(7-bromo-1-methyl-1H-indazol-3-yl)piperidine-2,6-dione 2913404-80-3 详细
tert-butyl N-[3-(3-oxoazetidin-1-yl)-1-bicyclo[1.1.1]pentanyl]carbamate 2654797-82-5 详细
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