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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
methyl 1-(morpholine-4-carbonyl)cyclopropanecarboxylate 1-(吗啉-4-羰基)环丙烷甲酸甲酯 1904338-15-3 详细
cis-2-(4-fluorophenyl)cyclopropanecarboxylic acid 950588-81-5 详细
(2R,7aS)-7a-[({4,7-dichloro-8-fluoropyrido[4,3-d]pyrimidin-2-yl}oxy)methyl]-2-fluoro-hexahydro-1H-pyrrolizine hydrochloride 详细
4-(2H-1,2,3,4-tetrazol-5-yl)piperidine hydrochloride 4-(2H-1,2,3,4-四唑-5-基)哌啶盐酸 91419-60-2 详细
1-cyclopropyl-1H-pyrazole-4-carboxylic acid 1-环丙基-1H-吡唑-4-羧酸 1622883-44-6 详细
tert-butyl 4-(4-bromo-1,3-thiazol-2-yl)piperazine-1-carboxylate 叔-丁基 4-(4-溴-1,3-噻唑-2-基)哌嗪-1-甲酸基酯 1197294-66-8 详细
2-chloro-7-cyclopentyl-N,N-dimethyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide 2-氯-7-环戊基-N,N-二甲基-7H-吡咯并[2,3-d]嘧啶-6-甲酰胺 1211443-61-6 详细
tert-butyl (3S)-4-(6-amino-3-pyridyl)-3-methyl-piperazine-1-carboxylate 1433849-58-1 1433849-58-1 详细
3-(4-methylphenyl)oxetan-3-yl]methanol 3-(4-甲基苯基)噁丁环烷-3-基]甲醇 1903050-29-2 详细
tert-butyl (4R)-2,2-dioxo-4-phenyl-1,2λ,3-oxathiazolidine-3-carboxylate 叔-丁基 (4R)-2,2-二氧亚基-4-苯基-1,2λ?,3-氧杂噻唑烷-3-甲酸基酯 1209467-60-6 详细
tert-butyl 4-[(azetidin-3-yl)(hydroxy)methyl]piperidine-1-carboxylate hydrochloride 4-(氮杂环丁烷-3-基(羟基)甲基)哌啶-1-羧酸叔丁酯盐酸盐 2227206-46-2 详细
trans-2-(3-fluoro-4-methoxy-phenyl)cyclopropanecarboxylic acid trans-2-(3-fluoro-4-methoxyphenyl)cyclopropane-1-carboxylic acid 1609290-12-1 详细
(6R)-6-(4-bromophenyl)-4-[(1S)-1-phenylethyl]morpholin-3-one 3-Morpholinone, 6-(4-bromophenyl)-4-[(1S)-1-phenylethyl]-, (6R)- 920801-93-0 详细
3-(1H-pyrazol-4-yl)cyclobutanamine dihydrochloride 详细
4-[1-(diphenylmethyl)azetidin-3-yl]morpholine 1-(DIPHENYLMETHYL)-3-(MORPHOLINO)AZETIDINE 55438-65-8 详细
(2S)-2-phenylpyrrolidine hydrochloride (2S)-2-苯基吡咯烷盐酸 56523-58-1 详细
3,3-dimethyl-1-[(1R)-1-phenylethyl]pyrrolidine-2,4-dione 3,3-二甲基-1-[(1R)-1-苯基乙基]吡咯烷-2,4-二酮 145704-80-9 详细
1-(4-Aminophenyl)cyclopentanecarbonitrile 1-(4-氨基苯基)环戊甲腈 115279-73-7 详细
2-bromo-6-(3-methoxytetrahydrofuran-3-yl)pyridine 2-溴-6-(3-甲氧基四氢呋喃-3-基)吡啶 2368946-64-7 详细
tert-butyl 3-indazol-1-ylpyrrolidine-1-carboxylate 2702457-70-1 详细
tert-butyl N-[(2R,3S)-2-(2,5-difluorophenyl)-5-oxooxan-3-yl]carbamate 叔-丁基 N-[(2R,3S)-2-(2,5-二氟苯基)-5-氧亚基噁烷-3-基]氨基甲酯 951127-25-6 详细
5-cyclopropyl-1-methyl-1H-imidazole-2-carboximidamide hydrochloride 5-环丙基-1-甲基-1H-咪唑-2-甲脒盐酸 1403766-70-0 详细
tert-butyl N-(4-phenylpiperidin-4-yl)carbamate 叔-丁基 N-(4-苯基哌啶-4-基)氨基甲酯 178914-47-1 详细
4-hydroxy-3,3-dimethyl-1-[(1R)-1-phenylethyl]pyrrolidin-2-one 4-羟基-3,3-二甲基-1-[(1R)-1-苯基乙基]吡咯烷-2-酮 1788065-51-9 详细
tert-butyl N-[trans-2-(4-hydroxyphenyl)cyclopropyl]carbamate 叔-丁基 N-[(1R,2S)-rel-2-(4-羟基苯基)环丙基]氨基甲酯 1196053-06-1 详细
1-(1-tert-butoxycarbonyl-4-piperidyl)cyclopropanecarboxylic acid 1-Boc-4-(1-carboxy-cyclopropyl)-piperidine 1363381-63-8 详细
1-[(benzyloxy)carbonyl]-3-phenylazetidine-3-carboxylic acid 1-[(苄氧基)羰基]-3-苯偶氮基丁啶-3-羧酸 1207203-37-9 详细
tert-butyl 4-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperazine-1-carboxylate 4-[4-(N-BOC)哌嗪-1-基]苯基硼酸频哪酯 470478-90-1 详细
4-(4-tert-butyl-2-ethoxyphenyl)-2-(2,6-difluorophenyl)-4,5-dihydro-1,3-oxazole 4-(4-叔-丁基-2-乙氧苯基)-2-(2,6-二氟苯基)-4,5-二氢-1,3-噁唑 153233-91-1 详细
3-(2-thienyl)azetidine;hydrochloride 2940950-45-6 详细
4-[4-(trifluoromethoxy)phenoxy]piperidine 4-[4-(三氟甲氧基)苯氧基]哌啶 287952-67-4 详细
4-(2-chlorothieno[3,2-d]pyrimidin-4-yl)morpholine 4-{2-氯噻吩并[3,2-d]嘧啶-4-基}吗啉 16234-15-4 详细
2,5-dichloro-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine 2,5-二氯-N-(5-甲基-1H-吡唑-3-基)嘧啶-4-胺 543712-81-8 详细
4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-ylsulfonyl)morpholine 4-(5-(4,4,5,5-四甲基-1,3,2-二氧杂环戊硼烷-2-基)吡啶-3-基磺酰基)吗啉 1093819-54-5 详细
3-(2-chloropyrimidin-4-yl)-1H-indole 3-(2-氯-嘧啶-4-基)-1H-吲哚 945016-63-7 详细
1-(4-bromophenyl)cyclobutanol 1-(4-溴苯基)环丁醇 19936-14-2 详细
(3S,4S)-4-(4-bromophenoxy)tetrahydrofuran-3-amine (3S,4S)-4-(4-bromophenoxy)tetrahydrofuran-3-amine 1258963-53-9 详细
3-pyrrolidin-1-ylcyclobutanamine;dihydrochloride 3-(吡咯烷-1-基)环丁胺二盐酸盐 1229625-04-0 详细
(4R,5R)-5-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-oxazolidin-2-one (4R,5R)-5-[3,5-双(三氟甲基)苯基] -4-甲基-1,3-噁唑烷-2-酮 875444-05-6 详细
5-[(3R)-3-methylmorpholin-4-yl]pyridin-2-amine 2-Pyridinamine, 5-[(3R)-3-methyl-4-morpholinyl]- 2375165-11-8 详细
(R)-phenyl-[(2S)-pyrrolidin-2-yl]methanol (ΑS, 2R)-Α-苯基-2-吡咯甲醇 74936-95-1 详细
(3R)-3-(5-bromo-1-oxo-isoindolin-2-yl)piperidine-2,6-dione (R)-3-(5-溴-1-氧异喹啉-2-基)哌啶-2,6-二酮 2243825-20-7 详细
trans-1-bromo-4-(3-fluorocyclobutyl)benzene 2954727-39-8 详细
1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-5-iodo-6-methyl-pyrimidine-2,4-dione 1-{[2-氟-6-(三氟甲基)苯基]甲基}-5-碘-6-甲基-1,2,3,4-四氢嘧啶-2,4-二酮 1150560-54-5 详细
3-phenyloxetane-3-carboxylic acid 3-苯基噁丁环烷-3-羧酸 114012-42-9 详细
4-(azetidin-1-yl)-4-phenylcyclohexan-1-one 4-(吖丁啶-1-基)-4-苯基环己烷-1-酮 1002916-47-3 详细
4-cyclopropyl-1H-imidazole-2-carbonitrile hydrochloride 4-环丙基-1H-咪唑-2-甲腈盐酸 2173991-69-8 详细
(2-(piperidin-1-yl)phenyl)boronic acid 2-哌啶基苯硼酸 1050505-85-5 详细
N,N-dimethyl-1-[3-(4-piperidyl)phenyl]methanamine;dihydrochloride 2244088-27-3 2244088-27-3 详细
1-[[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methyl]piperidine 1-{[4-(四甲基-1,3,2-二噁硼戊环-2-基)苯基]甲基}哌啶 859833-22-0 详细
{4-[1-(propan-2-yl)-4-(trifluoromethyl)-1H-imidazol-2-yl]phenyl}methanol 4-[1-异丙基-4-(三氟甲基)-2-咪唑基]苯基]甲醇 2446484-53-1 详细
N-[3-[[2-chloro-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]prop-2-enamide N-(3-{[2-氯-5-(三氟甲基)嘧啶-4-基]氨基}苯基)丙-2-烯酰胺 1374507-25-1 详细
4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)benzoic acid hydrochloride 4-[(4-乙基哌嗪-1-基)甲基]-3-(三氟甲基)苯甲酸盐酸 887565-40-4 详细
4'-Trifluoromethyl-biphenyl-4-carbaldehyde 4'-三氟甲基二苯基-4-甲醛 90035-34-0 详细
4-(aminomethyl)-4-fluoro-1-piperidyl]-(3-chloro-4-fluoro-phenyl)methanone;hydrochloride 1-[1-(3-氯-4-氟苯甲酰)-4-氟哌啶-4-基]甲胺盐酸 2173992-07-7 详细
5-[4-(trifluoromethyl)phenyl]morpholin-3-one 5-[4-(三氟甲基)苯基]吗啉-3-酮 1391087-84-5 详细
tert-butyl 3-(1H-triazol-5-yl)azepane-1-carboxylate 3-(1H-1,2,3-三唑-5-基)氮杂环庚烷-1-甲酸叔丁酯 2384722-09-0 详细
tert-butyl 4-[4-(methylamino)pyrazol-1-yl]piperidine-1-carboxylate 2504240-17-7 详细
tert-butyl trans-4-[(4-aminocyclohexyl)methyl]piperazine-1-carboxylate 1448362-67-1 详细
tert-butyl trans-3-(2,6-dichloropyridine-4-carbonyl)cyclobutanecarboxylate 2708283-76-3 详细
2-(1H-1,2,3-triazol-1-yl)benzoic acid 2-(1H-1,2,3-三唑-1-基)苯甲酸 1085458-53-2 详细
3-(2-chloropyrimidin-4-yl)-1-methyl-1H-indole 3-(2-氯嘧啶-4-基)-1-甲基-1H-吲哚 1032452-86-0 详细
tert-butyl (3S)-3-(4-aminophenyl)piperidine-1-carboxylate (3S)-3-(4-氨基苯基)哌啶-1-羧酸叔丁酯 1171197-20-8 详细
1-(benzothiophen-4-yl)piperazine;dihydrochloride 1-(1-苯并噻吩-4-基)哌嗪盐酸 1677681-05-8 详细
trans-2-(4-ethoxy-3-fluoro-phenyl)cyclopropanecarboxylic acid (1S,2S)-rel-2-(4-乙氧基-3-氟苯基)环丙烷-1-羧酸 2055840-75-8 详细
4-(3-chlorophenyl)-4-(dimethylamino)cyclohexan-1-one 65619-53-6 详细
6-oxo-1-phenyl-1,6-dihydropyridine-3-carboxylic acid 6-氧代-1-苯基-1,6-二氢吡啶-3-甲酸 77837-08-2 详细
2-(4-bromophenyl)-4H-1,2,4-triazol-3-one 2-(4-溴苯基)-1H-1,2,4-三唑-3(2H)-酮 197074-69-4 详细
(2R)-2-(4-bromophenyl)-4-[(1S)-1-phenylethyl]morpholine Morpholine, 2-(4-bromophenyl)-4-[(1S)-1-phenylethyl]-, (2R)- 920802-43-3 详细
2-(2-thienyl)piperazine 2-(2-噻吩基)]哌嗪 85803-49-2 详细
1-(4-methylpiperazin-1-yl)cyclopropanecarboxylic acid;dihydrochloride 2484905-94-2 详细
5-(azetidin-3-yl)-2-methyl-pyridine;dihydrochloride 2940940-62-3 详细
(4R)-4-phenylthiazolidine-2-thione (4R)-4-苯基-1,3-噻唑烷-2-硫酮 110199-18-3 详细
4-(1H-Pyrazol-4-yl)-7-((2-(trimethylsilyl)ethoxy)-methyl)-7H-pyrrolo[2,3-d]pyrimidine 4-(1H-吡唑-4-基)-7-((2-(三甲基硅烷基)乙氧基)-甲基)-7H-吡咯并[2,3-D]嘧啶 941685-27-4 详细
5-phenoxy-1,3-dihydro-2-benzofuran-1-one 5-苯氧基异苯并呋喃-1-(3H)-酮 57830-14-5 详细
2-chloro-4-cyclopropylpyridine 2-氯-4-环丙基吡啶 168975-75-5 详细
2-chloro-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid 2-氯-7-环戊基-7H-吡咯并[2,3-D]嘧啶-6-甲酸 1211443-58-1 详细
methyl 1-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]cyclopropane-1-carboxylate 甲基 4-(1-乙氧基羰基环丙基)苯硼酸频哪醇酯 1396007-85-4 详细
3-(4-chlorophenyl)oxetan-3-yl]methanol 3-(4-氯苯基)噁丁环烷-3-基]甲醇 1903083-49-7 详细
(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02]nona-1(6),7-diene-7-carboxylic acid (2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02]nona-1(6),7-diene-7-carboxylic acid 1268883-00-6 详细
4-(4-chloro-3-isopropyl-pyrazolo[3,4-b]pyridin-1-yl)-3-ethyl-benzonitrile 4-(4-氯-3-异丙基-1H-吡唑并[3,4-B]吡啶-1-基)-3-乙基苯甲腈 2306262-57-5 详细
1-(4-bromophenyl)cyclopropanesulfinic acid;sodium salt 2891599-32-7 详细
2-bromo-5-phenyl-1,3,4-oxadiazole 2-溴-5-苯基-1,3,4-噁二唑 51039-53-3 详细
tert-butyl N-[1-(4-aminophenyl)azetidin-3-yl]carbamate 叔-丁基 N-[1-(4-氨基苯基)吖丁啶-3-基]氨基甲酯 889948-10-1 详细
4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidin-2-yl)morpholine 2-(4-吗啡啉基)嘧啶-5-硼酸嚬哪醇酯 957198-30-0 详细
cis-4-phenylcyclohexanol 4α-Phenylcyclohexan-1α-ol 7335-12-8 详细
(3R)-3-(4-chlorophenyl)piperidine 1335689-11-6 1335689-11-6 详细
6-(4-oxopiperidin-1-yl)pyridine-3-carbonitrile 6-(4-氧亚基哌啶-1-基)吡啶-3-甲腈 116248-07-8 详细
4-{2-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]ethyl}morpholine 4-{2-[4-(四甲基-1,3,2-二噁硼戊环-2-基)-1H-吡唑-1-基]乙基}吗啉 864754-18-7 详细
4-(oxetan-3-yl)piperidine;hydrochloride 4-(氧杂环丁烷-3-基)哌啶盐酸盐 2648948-73-4 详细
tert-butyl (3S)-cis-4-(4-aminocyclohexyl)-3-(methoxymethyl)piperazine-1-carboxylate 2891581-08-9 详细
2-(morpholin-4-yl)pyrimidin-5-amine 2-(吗啉-4-基)嘧啶-5-胺 65735-68-4 详细
2-fluoro-5-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]benzoic acid 2-氟-5-[(4-氧亚基-3,4-二氢酞嗪-1-基)甲基]苯甲酸 763114-26-7 详细
ethenyldiphenylsulfanium trifluoromethanesulfonate 三氟甲磺酸化乙烯基二苯基硫烷正离子 247129-88-0 详细
6-cyclopropyl-3-nitro-pyridin-2-amine 6-cyclopropyl-3-nitro-pyridin-2-amine 1552286-03-9 详细
1-chloro-2-(chlorodiphenylmethyl)benzene 氯代(邻氯苯基)二苯基甲烷 42074-68-0 详细
2-(2,6-dioxo-3-piperidyl)-5-piperazin-1-yl-isoindoline-1,3-dione;hydrochloride 2-(2,6-二氧代哌啶-3-基)-5-(哌嗪-1-基)-2,3-二氢-1H-异吲哚-1,3-二酮盐酸盐 2228029-82-9 详细
methyl trans-4-[5-(difluoromethyl)-4-nitro-pyrazol-1-yl]cyclohexanecarboxylate 反式-4-[5-(二氟甲基)-4-硝基-1H-吡唑-1-基]环己烷羧酸甲酯 2434852-20-5 详细
3-phenylbicyclo[1.1.1]pentan-1-amine hydrobromide 3-苯基二环[1.1.1]戊烷-1-胺氢溴酸盐 1818847-90-3 详细
tert-butyl 4-fluoro-4-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperidine-1-carboxylate 1374342-20-7 详细
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