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PROTAC ER Degrader-4
- CAS No.
- 2361114-15-8
- Chemical Name:
- PROTAC ER Degrader-4
- Synonyms
- PROTAC ER Degrader-4
- CBNumber:
- CB28054603
- Molecular Formula:
- C53H67F3N6O8S
- Molecular Weight:
- 1005.19
- MDL Number:
- MFCD34469813
- MOL File:
- Mol file
Last updated:2024-07-02 08:55:04
PROTAC ER Degrader-4 Chemical Properties,Uses,Production
Biological Activity
PROTAC ER Degrader-4 is a von Hippel-Lindau-based PROATC estrogen receptor (ER) degrader, binding to ER with an IC50 of 0.8 nM. PROTAC ER Degrader-4 induces ER degradation in MCF-7 cells with an IC50 of 0.3 nM[1]. PROTAC ER Degrader-4 shows equal to 100% ER degradation at 0.3 μM in the MCF-7 ER degradation cellular assay[1].
References
[1]. Bin Yang, et al. Compounds and their use in treating cancer. WO2019123367A1.
PROTAC ER Degrader-4 Preparation Products And Raw materials
Raw materials
Preparation Products
PROTAC ER Degrader-4 Suppliers
Global( 5)Suppliers
Supplier | Tel | Country | ProdList | Advantage | |
---|---|---|---|---|---|
TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 | marketing@targetmol.com | United States | 19892 | 58 |
Sichuan Wei Keqi Biological Technology Co., Ltd. | 028-81700200 18116577057 | 3003855609@qq.com | China | 7887 | 56 |
Shanghai Chaolan Chemical Technology Center | QQ:65489617 15618227136 | info@SuperLan-chem.com | China | 9909 | 58 |
Jilin Province Woda Biotechnology Co., Ltd. | 13504435624 | 1927928688@qq.com | China | 1382 | 58 |
Changzhou Bojia Biomedical Technology Co., Ltd. | 2122619822 | czbjpharma@126.com | China | 18488 | 58 |
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PROTAC ER Degrader-4
2361114-15-8