Azamulin
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- ₹20069.55 - ₹78351.35
- Product name: Azamulin
- CAS: 76530-44-4
- MF: C24H38N4O4S
- MW: 478.65
- EINECS:
- MDL Number:MFCD00865055
- Synonyms:SA 85530b;14-O-(5-(2-Amino1,3,4-triazolyl)thioacetyl)dihydromutilin;Antibiotic TDM 85-530;Azamulin;[(5-Amino-1H-1,2,4-triazol-3-yl)thio]acetic acid (3aS,4R,5S,6R,8R,9R,9aR,10R)-6-ethyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester;TMD 85-530, SA 85530b;Acetic acid, 2-[(3-amino-1H-1,2,4-triazol-5-yl)thio]-, (3aS,4R,5S,6R,8R,9R,9aR,10R)-6-ethyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester
2 prices
Selected condition:
Brand
- Sigma-Aldrich(India)
Package
- 5MG
- 25MG
- ManufacturerSigma-Aldrich(India)
- Product numberSML0485
- Product descriptionAzamulin ≥98% (HPLC)
- Packaging5MG
- Price₹20069.55
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberSML0485
- Product descriptionAzamulin ≥98% (HPLC)
- Packaging25MG
- Price₹78351.35
- Updated2022-06-14
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
Sigma-Aldrich(India) | SML0485 | Azamulin ≥98% (HPLC) | 5MG | ₹20069.55 | 2022-06-14 | Buy |
Sigma-Aldrich(India) | SML0485 | Azamulin ≥98% (HPLC) | 25MG | ₹78351.35 | 2022-06-14 | Buy |
Properties
Melting point :128-130°C
Boiling point :659.4±65.0 °C(Predicted)
Density :1.27±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL (clear solution)
form :powder
pka :9.56±0.40(Predicted)
color :white to beige
Stability :Store at -2℃.
Boiling point :659.4±65.0 °C(Predicted)
Density :1.27±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL (clear solution)
form :powder
pka :9.56±0.40(Predicted)
color :white to beige
Stability :Store at -2℃.
Safety Information
Symbol(GHS): |
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Signal word: | Warning | ||||||||||||||||||||||||||||
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Description
Azamulin is a selective, irreversible inhibitor of cytochrome P450 (CYP) 3A isoforms (IC50 values range from 26 to 240 nM for CYP3A4 and CYP3A4/5 from different sources). It is at least 50-fold less potent against CYP2J2 and 100-fold less effective against all other CYP isoforms. Azamulin potently blocks the hydroxylation of testosterone and midazolam by CYP3A4.Related product price
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