Elacridar
- ₹9600 - ₹62038.08
- Product name: Elacridar
- CAS: 143664-11-3
- MF: C34H33N3O5
- MW: 563.64
- EINECS:1532714-185-1
- MDL Number:MFCD00912604
- Synonyms:elacridar;n-[4-[2-(6,7-dimethoxy-3,4-dihydro-1h-isoquinolin-2-yl)ethyl]phenyl]-5-methoxy-9-oxo-10h-acridine-4-carboxamide;GF 120918;GG 918;GW 0918;N-[4-[2-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]-9,10-dihydro-5-methoxy-9-oxo-4-acridinecarboxamide;N-[4-[2-(3,4-Dihydro-6,7-diMethoxy-isoquinolin-2(1H)-yl)ethyl]phenyl]-9,10-dihydro-5-Methoxy-9-oxo-4-acridinecarboxaMide;1-{2-carbaMoyl-5-[2-(6,7-diMethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]phenyl}-5-Methoxy-9-oxo-9,10-dihydroacridine-4-carboxylic acid
4 prices
Selected condition:
Brand
- TCI Chemicals (India)
- Sigma-Aldrich(India)
Package
- 10MG
- 25MG
- 50MG
- 100MG
- ManufacturerTCI Chemicals (India)
- Product numberE1371
- Product descriptionElacridar
- Packaging25MG
- Price₹9600
- Updated2022-05-26
- Buy
- ManufacturerTCI Chemicals (India)
- Product numberE1371
- Product descriptionElacridar
- Packaging100MG
- Price₹23100
- Updated2022-05-26
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberSML0486
- Product descriptionElacridar ≥98% (HPLC)
- Packaging10MG
- Price₹15403.98
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberSML0486
- Product descriptionElacridar ≥98% (HPLC)
- Packaging50MG
- Price₹62038.08
- Updated2022-06-14
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
TCI Chemicals (India) | E1371 | Elacridar | 25MG | ₹9600 | 2022-05-26 | Buy |
TCI Chemicals (India) | E1371 | Elacridar | 100MG | ₹23100 | 2022-05-26 | Buy |
Sigma-Aldrich(India) | SML0486 | Elacridar ≥98% (HPLC) | 10MG | ₹15403.98 | 2022-06-14 | Buy |
Sigma-Aldrich(India) | SML0486 | Elacridar ≥98% (HPLC) | 50MG | ₹62038.08 | 2022-06-14 | Buy |
Properties
Melting point :216-218°C
Boiling point :701.6±60.0 °C(Predicted)
Density :1.264±0.06 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: soluble2mg/mL (clear solution, warmed)
form :powder
pka :12.58±0.70(Predicted)
color :white to beige
CAS DataBase Reference :143664-11-3(CAS DataBase Reference)
Boiling point :701.6±60.0 °C(Predicted)
Density :1.264±0.06 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: soluble2mg/mL (clear solution, warmed)
form :powder
pka :12.58±0.70(Predicted)
color :white to beige
CAS DataBase Reference :143664-11-3(CAS DataBase Reference)
Safety Information
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Signal word: | Warning | ||||||||||||||
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Description
Elacridar is a dual inhibitor of P-glycoprotein (MRP-1, ABCB1) and breast cancer resistance protein (BCRP, ABCG2). It maximally inhibits P-glycoprotein in isolated human peripheral blood leukocytes at 200 nM. Elacridar blocks the activity of P-glycoprotein at the blood-brain barrier, altering the pharmacokinetics of certain drugs in the brain. This compound is effective against both human BCRP and the mouse homolog, Bcrp1.Related product price
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