Enzastaurin (LY317615)
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- ₹11506.98 - ₹46374.3
- Product name: Enzastaurin (LY317615)
- CAS: 170364-57-5
- MF: C32H29N5O2
- MW: 515.6
- EINECS:
- MDL Number:MFCD11040980
- Synonyms:1H-Pyrrole-2,5-dione, 3-(1-methyl-1H-indol-3-yl)-4-(1-(1-(2-pyridinylmethyl)-4-piperidinyl)-1H-indol-3-yl)-;Unii-uc96G28eqf;Enzastaurin,Enzstataurin,LY317615,170364-57-5,1H-Pyrrole-2,5-dione, 3-;3-(1-Methyl-1H-indol-3-yl)-4-(1-(1-(2-pyridinylmethyl)-4-piperidinyl)-1H-indol-3-yl)-1H-pyrrole-2,5-dione;Enzastaurin ( LY317615 );Enzastaurine;LY317615 (Enzastaurin);LY317615/Enzstataurin
2 prices
Selected condition：
Brand
- Sigma-Aldrich(India)
Package
- 5MG
- 25MG
- ManufacturerSigma-Aldrich(India)
- Product numberSML0762
- Product descriptionEnzastaurin ≥98% (HPLC)
- Packaging5MG
- Price₹11506.98
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberSML0762
- Product descriptionEnzastaurin ≥98% (HPLC)
- Packaging25MG
- Price₹46374.3
- Updated2022-06-14
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Sigma-Aldrich(India) | SML0762 | Enzastaurin ≥98% (HPLC) | 5MG | ₹11506.98 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | SML0762 | Enzastaurin ≥98% (HPLC) | 25MG | ₹46374.3 | 2022-06-14 | Buy |
Properties
Melting point :249-261℃
Boiling point :767.2±60.0 °C(Predicted)
Density :1.34
RTECS :UX9626850
Flash point :417.8℃
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL, clear (warmed)
form :powder
pka :7.88±0.60(Predicted)
color :, light orange to dark orange-red
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Boiling point :767.2±60.0 °C(Predicted)
Density :1.34
RTECS :UX9626850
Flash point :417.8℃
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL, clear (warmed)
form :powder
pka :7.88±0.60(Predicted)
color :, light orange to dark orange-red
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
Enzastaurin is a potent inhibitor of PKCβ (IC50 = 6 nM), with modest selectivity over PKCα, PKCγ, and PKCε (IC50 = 39, 83, and 110 nM, respectively). At 3 μM, enzastaurin also inhibits signaling through the Akt pathway. It suppresses angiogenesis, induces apoptosis, and reduces proliferation of cultured tumor cells. Because of these effects, enzastaurin has potential antineoplastic activity.More related product prices
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