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Rilmenidine

CAS No.: 54187-04-1

Chemical Name:: Rilmenidine

Synonyms: s3341;Tenaxum;Hyperium;S-3341-3;RILMENIDINE;oxaminozoline;TENAXUM; HYPERIUM;Rilmenidine USP/EP/BP;Rilmenidinehemifuramate;RilMenidine heMifuMarate sa

CBNumber:: CB0391076

Molecular Formula:: C10H16N2O

Molecular Weight:: 180.25

MOL File:: 54187-04-1.mol

MSDS File:: SDS

Modify Date:: 2024/5/30 16:33:02

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Rilmenidine Properties

Melting point	106-107°
Boiling point	355.5±9.0 °C(Predicted)
Density	1.45±0.1 g/cm3(Predicted)
storage temp.	Store at -20°C
solubility	H₂O: 7.3 mg/mL
form	solid
pka	7.88±0.50(Predicted)
color	white
CAS DataBase Reference	54187-04-1(CAS DataBase Reference)

SAFETY

Risk and Safety Statements

Safety Statements	22-24/25
WGK Germany	3
RTECS	RP7207400

Rilmenidine Chemical Properties,Uses,Production

Description

Rilmenidine is a new antihypertensive agent with a selective alphaz-agonist/antagonist profile, reportedly useful in the management of mild to moderate hypertension. Its fmt-line indication is possible because of the clear dissociation of its antihypertensive activity from other neurophannacological effects.

Chemical Properties

water soluble

Uses

I1-imidazoline binding site ligand and a2-adrenoceptor agonist, exhibits higher I1 vs. a2 selectivity than clonidine

Biological Activity

I 1 -imidazoline binding site selective ligand and α 2 -adrenoceptor agonist. Possesses greater I 1 vs α 2 selectivity than the prototypical compound, clonidine.

Metabolic pathway

In short-term rat hepatocyte cultures, oxaminozoline is metabolized and its four metabolites resulting from oxidation or hydrolysis are identified, three of which are identical to those reported in vivo. The presence of an additional minor metabolite in culture may be due to the higher metabolic rate of oxaminozoline in this model system.

Rilmenidine Preparation Products And Raw materials

Raw materials

Monoethanolamine Phenyl chloroformate 2-Chloroethyl isocyanate Thionyl chloride

Preparation Products

Rilmenidine Suppliers

Global( 131)Suppliers

Supplier	Tel	Country	ProdList	Advantage	Inquiry
Varanous Labs Pvt Ltd	+91-7036248882 +91-7036248882	Hyderabad, India	1541	58	Inquiry
CLEARSYNTH LABS LTD.	+91-22-45045900	Hyderabad, India	6351	58	Inquiry
Pharmaffiliates Analytics and Synthetics P. Ltd	+91-172-5066494	Haryana, India	6773	58	Inquiry
Hebei Duling International Trade Co. LTD	+8617333973358	China	15438	58	Inquiry
CONIER CHEM AND PHARMA LIMITED	+8618523575427	China	49391	58	Inquiry
SIMAGCHEM CORP	+86-13806087780	China	17367	58	Inquiry
Hefei TNJ Chemical Industry Co.,Ltd.	0551-65418671	China	34571	58	Inquiry
Shaanxi Dideu Medichem Co. Ltd	+86-029-89586680 +86-18192503167	China	9030	58	Inquiry
AFINE CHEMICALS LIMITED	+86-0571-85134551	China	15395	58	Inquiry
Baoji Guokang Healthchem co.,ltd	+8615604608665 15604608665	CHINA	9427	58	Inquiry

Supplier	Advantage
Varanous Labs Pvt Ltd	58
CLEARSYNTH LABS LTD.	58
Pharmaffiliates Analytics and Synthetics P. Ltd	58
Hebei Duling International Trade Co. LTD	58
CONIER CHEM AND PHARMA LIMITED	58
SIMAGCHEM CORP	58
Hefei TNJ Chemical Industry Co.,Ltd.	58
Shaanxi Dideu Medichem Co. Ltd	58
AFINE CHEMICALS LIMITED	58
Baoji Guokang Healthchem co.,ltd	58

54187-04-1(Rilmenidine)Related Search:

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(S)-1-CYCLOPROPYLETHYLAMINE RILMENIDINE DIHYDROGEN PHOSPHATE,rilmenidine phosphate O-METHYLISOUREA ACETATE RILMENIDINE FOR SYSTEM SUITABILITY Oxazoline

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n-(dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine oxaminozoline RILMENIDINE 1,1-dicyclopropyl-n-(2-oxazolinyl)-methylamin 2-((dicyclopropylmethyl)imino)-oxazolidin 2-((dicyclopropylmethyl)imino)oxazolidine 2-(dicyclopropylmethylamino)-2-oxazoline 4,5-dihydro-n-(dicyclopropylmethyl)-2-oxazolamin s3341 N-(dicyclopropylmethyl)-4,5-dihydrooxazol-2-amine 2-(N-(Dicyclopropylmethyl)amino)oxazolinehemifuramate Rilmenidinehemifuramate Rilmenidine 2-[(Dicyclopropylmethyl)amino]-2-oxazoline Hyperium S-3341-3 RilMenidine heMifuMarate sa 2-[N-(Dicyclopropylmethyl)amino]oxazoline fumarate (2:1) salt N-(2-Oxazolin-2-yl)-α,α-dicyclopropylmethanamine Oxaminozoline hemifumarate salt Rilmenidene hemifumarate salt RilmenidineQ: What is Rilmenidine Q: What is the CAS Number of Rilmenidine Q: What is the storage condition of Rilmenidine Rilmenidine USP/EP/BP 2-Oxazolamine, N-(dicyclopropylmethyl)-4,5-dihydro- TENAXUM; HYPERIUM Tenaxum N-(dicyclopropyl methyl)-4, 5-dihydro2-oxazolamide 54187-04-1 54178-04-1 C10H16N2OC4H4O4 C10H16N2O05C4H4O4 C10H16N2O189C4H4O4 Antihypertensive Imidazoline binding site