ChemicalBook > Product Catalog >Biochemical Engineering >Inhibitors >protein tyrosine kinase >PELITINIB
PELITINIB
- CAS No.
- 257933-82-7
- Chemical Name:
- PELITINIB
- Synonyms
- Pelitinib(EKB-569);PELITINIB;WAY172569;WAY 172569;WAY-172569;WAY-EKB 569;Pelitinib, >=98%;EKB-569 Pelitinib;257933-82-7 PELITINIB;PELITINIB (EKB-569;WAY-EKB 569)
- CBNumber:
- CB81011748
- Molecular Formula:
- C24H23ClFN5O2
- Molecular Weight:
- 467.92
- MOL File:
- 257933-82-7.mol
- MSDS File:
- SDS
- Modify Date:
- 2023/6/30 15:45:59
PELITINIB price More Price(4)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich(India) | PZ0197 | Pelitinib ≥98% (HPLC) | 257933-82-7 | 5MG | ₹14440.55 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | PZ0197 | Pelitinib ≥98% (HPLC) | 257933-82-7 | 25MG | ₹58151.9 | 2022-06-14 | Buy |
| TCI Chemicals (India) | P2529 | Pelitinib | 257933-82-7 | 25MG | ₹8300 | 2022-05-26 | Buy |
| TCI Chemicals (India) | P2529 | Pelitinib | 257933-82-7 | 100MG | ₹14800 | 2022-05-26 | Buy |
PELITINIB Chemical Properties,Uses,Production
Description
Pelitinib is a cyanoquinoline that irreversibly inhibits the EGFR receptor tyrosine kinase (IC50 = 39 nM). It inhibits HER2 with a much weaker potency (IC50 = 1.2 μM). By disrupting Akt and MAPK pathways, pelitinib can induce apoptosis and suppress the growth of tumor cell lines, displaying particularly strong efficacy against hepatocellular carcinoma cells (IC50s = ~2 μM).
Chemical Properties
Off-White Solid
Uses
Labelled Pelitinib (P218702). A tyrosine kinase inhibitor; it is used to prepare formulation for treating primary or secondary cancer.
PELITINIB Preparation Products And Raw materials
Raw materials
Preparation Products
Global( 192)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | Inquiry |
|---|---|---|---|---|---|
| TCI Chemicals (India) Pvt. Ltd. | 1800 425 7889 | New Delhi, India | 6778 | 58 | Inquiry |
| A.J Chemicals | 91-9810153283 | New Delhi, India | 6124 | 58 | Inquiry |
| CLEARSYNTH LABS LTD. | +91-22-45045900 | Hyderabad, India | 6351 | 58 | Inquiry |
| Pharma Affiliates | 172-5066494 | Haryana, India | 6761 | 58 | Inquiry |
| Anant Pharmaceuticals Pvt. ltd | +91 8550986868 | Maharashtra, India | 736 | 58 | Inquiry |
| Pharmaffiliates Analytics and Synthetics P. Ltd | +91-172-5066494 | Haryana, India | 6773 | 58 | Inquiry |
| Capot Chemical Co.,Ltd. | 571-85586718 +8613336195806 | China | 29798 | 60 | Inquiry |
| Henan Tianfu Chemical Co.,Ltd. | +86-0371-55170693 +86-19937530512 | China | 21676 | 55 | Inquiry |
| ATK CHEMICAL COMPANY LIMITED | +undefined-21-51877795 | China | 32760 | 60 | Inquiry |
| career henan chemical co | +86-0371-86658258 +8613203830695 | China | 29901 | 58 | Inquiry |
257933-82-7(PELITINIB)Related Search:
chevron_left
1of3
chevron_right
PELITINIB
2-Butenamide, N-[4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-, (2E)-
(2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide
WAY-EKB 569
(2E)-N-{4-[(3-chloro-4-fluorophenyl)aMino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(diMethylaMino)but-2-enaMide
(E)-N-(4-(3-chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)but-2-enamide
(2e)-n-(4-((3-chloro-4-fluorophenyl)aMino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(diMethylaMino)-2-butenaMide pelitinib
N-[4-(3-Chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)-2(E)-but·Namide
EKB-569 Pelitinib
Pelitinib (2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide
Pelitinib, >=98%
(E)-N-(4-(3-Chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)but-2-
PELITINIB (EKB-569;WAY-EKB 569)
EKB-569; WAY-EKB 569; EKB569; EKB 569
257933-82-7 PELITINIB
Pelitinib(EKB-569)
WAY 172569
WAY172569
WAY-172569
257933-82-7
C24H23ClFN5O2
C24H17D6ClFN5O2
Inhibitors
Intermediates & Fine Chemicals
Pharmaceuticals
Tyrosine Kinase Inhibitors
pyridine
All Inhibitors
API
Aromatics
Heterocycles
Isotope Labelled Compounds