PELITINIB
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- ₹8300 - ₹58151.9
- Product name: PELITINIB
- CAS: 257933-82-7
- MF: C24H23ClFN5O2
- MW: 467.92
- EINECS:803-625-4
- MDL Number:MFCD09837868
- Synonyms:PELITINIB;2-Butenamide, N-[4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-, (2E)-;(2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide;WAY-EKB 569;(2E)-N-{4-[(3-chloro-4-fluorophenyl)aMino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(diMethylaMino)but-2-enaMide;(E)-N-(4-(3-chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)but-2-enamide;(2e)-n-(4-((3-chloro-4-fluorophenyl)aMino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(diMethylaMino)-2-butenaMide pelitinib;N-[4-(3-Chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)-2(E)-but·Namide
4 prices
Selected condition：
Brand
- TCI Chemicals (India)
- Sigma-Aldrich(India)
Package
- 5MG
- 25MG
- 100MG
- ManufacturerTCI Chemicals (India)
- Product numberP2529
- Product descriptionPelitinib
- Packaging25MG
- Price₹8300
- Updated2022-05-26
- Buy
- ManufacturerTCI Chemicals (India)
- Product numberP2529
- Product descriptionPelitinib
- Packaging100MG
- Price₹14800
- Updated2022-05-26
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberPZ0197
- Product descriptionPelitinib ≥98% (HPLC)
- Packaging5MG
- Price₹14440.55
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberPZ0197
- Product descriptionPelitinib ≥98% (HPLC)
- Packaging25MG
- Price₹58151.9
- Updated2022-06-14
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| TCI Chemicals (India) | P2529 | Pelitinib | 25MG | ₹8300 | 2022-05-26 | Buy |
| TCI Chemicals (India) | P2529 | Pelitinib | 100MG | ₹14800 | 2022-05-26 | Buy |
| Sigma-Aldrich(India) | PZ0197 | Pelitinib ≥98% (HPLC) | 5MG | ₹14440.55 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | PZ0197 | Pelitinib ≥98% (HPLC) | 25MG | ₹58151.9 | 2022-06-14 | Buy |
Properties
Melting point :173-178°C
Boiling point :655.5±55.0 °C(Predicted)
Density :1.34
storage temp. :Keep in dark place,Inert atmosphere,Store in freezer, under -20°C
solubility :DMSO: soluble5mg/mL, clear (warmed)
form :powder
pka :12.23±0.43(Predicted)
color :white to beige
Boiling point :655.5±55.0 °C(Predicted)
Density :1.34
storage temp. :Keep in dark place,Inert atmosphere,Store in freezer, under -20°C
solubility :DMSO: soluble5mg/mL, clear (warmed)
form :powder
pka :12.23±0.43(Predicted)
color :white to beige
Safety Information
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| Signal word: | Danger | ||||||||||||||
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Description
Pelitinib is a cyanoquinoline that irreversibly inhibits the EGFR receptor tyrosine kinase (IC50 = 39 nM). It inhibits HER2 with a much weaker potency (IC50 = 1.2 μM). By disrupting Akt and MAPK pathways, pelitinib can induce apoptosis and suppress the growth of tumor cell lines, displaying particularly strong efficacy against hepatocellular carcinoma cells (IC50s = ~2 μM).More related product prices
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₹18270-50200 - 4-[(3-BROMOPHENYL)AMINO]-6-ACRYLAMIDOQUINAZOLINE
₹11539.45-46547.5 - PELITINIB
₹8300-58151.9
