GF109203X
|
- ₹4000 - ₹88851.6
- Product name: GF109203X
- CAS: 133052-90-1
- MF: C25H24N4O2
- MW: 412.48
- EINECS:
- MDL Number:MFCD00236428
- Synonyms:Bisindolylmaleimide I (GF 109203X);InSolution? Bisindolylmaleimide I ;GO 6850;GO 6850 HCL;GF 109203X;GF-109203X HCL;GF109203X HYDROCHLORIDE;BISINDOLYLMALEIMIDE
8 prices
Selected condition：
Brand
- Sigma-Aldrich
- TCI Chemicals (India)
- Sigma-Aldrich(India)
Package
- 1MG
- 5MG
- 25MG
- 1ML
- 250μG
- ManufacturerSigma-Aldrich
- Product number203290
- Product descriptionBisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine.
- Packaging250μG
- Price₹7070
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich
- Product number203290
- Product descriptionBisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine.
- Packaging1MG
- Price₹19490.01
- Updated2022-06-14
- Buy
- ManufacturerTCI Chemicals (India)
- Product numberB5781
- Product descriptionBisindolylmaleimide I
- Packaging5MG
- Price₹4000
- Updated2022-05-26
- Buy
- ManufacturerTCI Chemicals (India)
- Product numberB5781
- Product descriptionBisindolylmaleimide I
- Packaging25MG
- Price₹12000
- Updated2022-05-26
- Buy
- ManufacturerSigma-Aldrich(India)
- Product number203290
- Product descriptionBisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine.
- Packaging250μG
- Price₹7070
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product number203290
- Product descriptionBisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine.
- Packaging1MG
- Price₹19490.01
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product number203293
- Product descriptionInSolution Bisindolylmaleimide I - CAS 133052-90-1 - Calbiochem
- Packaging1ML
- Price₹21460
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberG2911
- Product descriptionGF 109203X synthetic, ≥90% (HPLC)
- Packaging1MG
- Price₹88851.6
- Updated2022-06-14
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Sigma-Aldrich | 203290 | Bisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine. | 250μG | ₹7070 | 2022-06-14 | Buy |
| Sigma-Aldrich | 203290 | Bisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine. | 1MG | ₹19490.01 | 2022-06-14 | Buy |
| TCI Chemicals (India) | B5781 | Bisindolylmaleimide I | 5MG | ₹4000 | 2022-05-26 | Buy |
| TCI Chemicals (India) | B5781 | Bisindolylmaleimide I | 25MG | ₹12000 | 2022-05-26 | Buy |
| Sigma-Aldrich(India) | 203290 | Bisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine. | 250μG | ₹7070 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | 203290 | Bisindolylmaleimide I - CAS 133052-90-1 - Calbiochem A highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (IC?? = 10 nM) that is structurally similar to staurosporine. | 1MG | ₹19490.01 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | 203293 | InSolution Bisindolylmaleimide I - CAS 133052-90-1 - Calbiochem | 1ML | ₹21460 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | G2911 | GF 109203X synthetic, ≥90% (HPLC) | 1MG | ₹88851.6 | 2022-06-14 | Buy |
Properties
Melting point :280℃ (decomposition)
Boiling point :685.6±55.0 °C(Predicted)
Density :1.30±0.1 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: ~1 mg/mlsoluble
form :Liquid
pka :8.13±0.60(Predicted)
color :Orange
Water Solubility :Insoluble in water.
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 6 months.
Boiling point :685.6±55.0 °C(Predicted)
Density :1.30±0.1 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: ~1 mg/mlsoluble
form :Liquid
pka :8.13±0.60(Predicted)
color :Orange
Water Solubility :Insoluble in water.
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 6 months.
Safety Information
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| Signal word: | Danger | ||||||||||||||
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Description
Bisindolylmaleimide I (BIM I) is a highly selective, cell-permeable, and reversible protein kinase C (PKC) inhibitor (Ki = 14 nM) that is structurally similar to the poorly selective PKC inhibitor staurosporine. It acts as a competitive inhibitor for the ATP binding site of PKC and shows high selectivity for PKCα-, β1-, β2-, γ-, δ-, and ε-isozymes. BIM I directly inhibits GSK3 in primary adipocyte lysates (IC50 = 360 nM) and in GSK3β immunoprecipitates derived from rat epididymal adipocytes (IC50 = 170 nM). This compound also competitively antagonizes the 5-HT3 receptor with a Ki value of 61 nM.More related product prices
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- GF109203X
₹4000-88851.6 - Bisindolylmaleimide V
₹7070-22650 - 119139-23-0
₹5400-31121.88
