Tianeptine sodium salt
- CAS No.
- 30123-17-2
- Chemical Name:
- Tianeptine sodium salt
- Synonyms
- TIANEPTINE SODIUM;Tianeptine Free Acid;Stablon;S-1574;99% purity Tianeptine sodium salt;7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Acid S,S-Dioxide Sodium Salt;tianeptin sodium;Coaxil sodiuM salt;tianeptin-a sodium;Tianeptine Sodium SaL
- CBNumber:
- CB9279090
- Molecular Formula:
- C21H24ClN2NaO4S
- Molecular Weight:
- 458.93
- MOL File:
- 30123-17-2.mol
- MSDS File:
- SDS
- Modify Date:
- 2024/7/19 18:29:52
| Melting point | 1800C |
|---|---|
| storage temp. | Desiccate at RT |
| solubility | DMSO: ≥20mg/mL |
| form | solid |
| color | white to tan |
| Merck | 14,9420 |
| Stability | Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 2 months. |
| InChIKey | ZLBSUOGMZDXYKE-UHFFFAOYSA-M |
| SMILES | C1(NCCCCCCC([O-])=O)C2C=CC=CC=2N(C)S(=O)(=O)C2C=C(Cl)C=CC1=2.[Na+] |
| CAS DataBase Reference | 30123-17-2(CAS DataBase Reference) |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS07 |
|---|---|
| Signal word | Warning |
| Hazard statements | H302-H312-H332 |
| Precautionary statements | P261-P271-P304+P340-P312-P280-P302+P352-P312-P322-P363-P501-P264-P270-P301+P312-P330-P501 |
| WGK Germany | 3 |
| HS Code | 2934.99.4400 |
Tianeptine sodium salt price More Price(4)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich(India) | T1692 | Tianeptine sodium salt hydrate ≥98% (HPLC), powder | 30123-17-2 | 5MG | ₹28826.98 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | T1692 | Tianeptine sodium salt hydrate ≥98% (HPLC), powder | 30123-17-2 | 25MG | ₹114972.33 | 2022-06-14 | Buy |
| TCI Chemicals (India) | T3131 | Tianeptine Sodium Salt | 30123-17-2 | 200MG | ₹9200 | 2022-05-26 | Buy |
| TCI Chemicals (India) | T3131 | Tianeptine Sodium Salt | 30123-17-2 | 1G | ₹19800 | 2022-05-26 | Buy |
Tianeptine sodium salt Chemical Properties,Uses,Production
Description
Tianeptine sodium salt is a structurally novel, serotonin specific antidepressant. It is useful in the treatment of neurotic and reactive depressions, as well as depressive states accompanied by anxiety. Tianeptine (sodium salt) is an analytical reference standard categorized as an opioid. Tianeptine has been abused and associated with overdose and death. Formulations containing tianeptine have been used in the treatment of depression. This product is intended for use in analytical forensic applications. This product is also available as a general research tool .
Uses
Tianeptine sodium salt is a tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. Tianeptine sodium salt hydrate has been used as a selective serotonin reuptake enhancer (SSRE) positive control during serotonin transporter (SERT) assay in human embryonic kidney 293 cell lines. Tianeptine (INN) (Stablon, Coaxil, Tatinol) is a SSRE drug used for treating major depressive episodes (mild, moderate, or severe). Tianeptine commonly used for depression. It is also used for pain, asthma, anxiety, and many other conditions, but there is no good scientific evidence to support these other uses.
General Description
Tianeptine is a μ-opioid receptor (MOR) as well as a δ-opioid receptor (DOR) agonist.
Biological Activity
Selective facilitator of 5-HT uptake in vitro and in vivo . Has no affinity for a wide range of receptors, including 5-HT and dopamine (IC 50 > 10 μ M) and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo .
Tianeptine sodium salt Preparation Products And Raw materials
| Supplier | Tel | Country | ProdList | Advantage | Inquiry |
|---|---|---|---|---|---|
| Bulat Pharmaceutical Pvt Ltd | +91-8448085659 +91-8448085660 | Haryana, India | 123 | 58 | Inquiry |
| Ralington Pharma | +91-7948911722 +91-9687771722 | Gujarat, India | 1350 | 58 | Inquiry |
| CLEARSYNTH LABS LTD. | +91-22-45045900 | Hyderabad, India | 6351 | 58 | Inquiry |
| A.J Chemicals | 91-9810153283 | New Delhi, India | 6124 | 58 | Inquiry |
| TCI Chemicals (India) Pvt. Ltd. | 1800 425 7889 | New Delhi, India | 6778 | 58 | Inquiry |
| Pharmaffiliates Analytics and Synthetics P. Ltd | +91-172-5066494 | Haryana, India | 6773 | 58 | Inquiry |
| SynZeal Research Pvt Ltd | +1 226-802-2078 | Gujarat, India | 6522 | 58 | Inquiry |
| Neel Kanth Drugs Private Limited | 08069033721Ext 594 | Delhi, India | 6 | 58 | Inquiry |
| Neuland Laboratories Limited | +91 40 67611600 / 1700 | New Delhi, India | 2 | 58 | Inquiry |
| Prasol Chemicals Private Limited | 08046048267 | Mumbai, India | 49 | 58 | Inquiry |
Related articles
- Synthesis and Biological Activity of Tianeptine sodium salt
- Tianeptine sodium salt not only has good antidepressant effect, but also has fewer adverse reactions than traditional tricycli....
- Jul 20，2022
Related Qustion
- Q:What is the biological activity of Tianeptine sodium salt?
- A:Tianeptine sodium salt (TSS) is a facilitator of serotonin and norepinephrine reuptake.
- Sep 9，2024
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