Eliprodil
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- ₹7470 - ₹60100
- Product name: Eliprodil
- CAS: 119431-25-3
- MF: C20H23ClFNO
- MW: 347.85
- EINECS:
- MDL Number:MFCD00866651
- Synonyms:SL 820715;ALPHA-(4-CHLOROPHENYL)-4-[(4-FLUOROPHENYL)METHYL]-1-PIPERIDINEETHANOL;ELIPRODIL;α-(4-chlorophenyl)-4-[(4-fluorophenyl)methyl]-1-piperidineethanol;SL 820715, α-(4-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1-piperidineethanol;(+-)-alpha-(p-Chlorophenyl)-4-(p-fluorobenzyl)-1-piperidineethanol;1-(4-broMophenyl)-2-(4-(4-fluorobenzyl)piperidin-1-yl)ethanol;1-Piperidineethanol, α-(4-chlorophenyl)-4-[(4-fluorophenyl)methyl]-
3 prices
Selected condition：
Brand
- Sigma-Aldrich(India)
Package
- 10MG
- 50MG
- ManufacturerSigma-Aldrich(India)
- Product number5.04539
- Product descriptionEliprodil - CAS 119431-25-3 - Calbiochem
- Packaging10MG
- Price₹7470
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberE2031
- Product descriptionEliprodil ≥98% (HPLC), powder
- Packaging10MG
- Price₹13350
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberE2031
- Product descriptionEliprodil ≥98% (HPLC), powder
- Packaging50MG
- Price₹60100
- Updated2022-06-14
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Sigma-Aldrich(India) | 5.04539 | Eliprodil - CAS 119431-25-3 - Calbiochem | 10MG | ₹7470 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | E2031 | Eliprodil ≥98% (HPLC), powder | 10MG | ₹13350 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | E2031 | Eliprodil ≥98% (HPLC), powder | 50MG | ₹60100 | 2022-06-14 | Buy |
Properties
Boiling point :474.1±35.0 °C(Predicted)
Density :1.205±0.06 g/cm3(Predicted)
storage temp. :Sealed in dry,2-8°C
solubility :DMSO: ~17 mg/mL
form :solid
pka :13.99±0.20(Predicted)
color :white
Density :1.205±0.06 g/cm3(Predicted)
storage temp. :Sealed in dry,2-8°C
solubility :DMSO: ~17 mg/mL
form :solid
pka :13.99±0.20(Predicted)
color :white
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
N-Methyl-D-aspartate (NMDA) receptors are calcium permeable ligand-gated channels of the central nervous system that are activated after binding of the co-agonists glutamate and glycine. Eliprodil is a non-competitive NMDA receptor antagonist that inhibits neuronal calcium channel currents. It is selective for NR2B subunit-containing receptors (IC50 = 1 μM), displaying greater than 100-fold selectivity for NR2B over NR2A and NR2C subunits. Eliprodil also avidly binds σ1 and σ2 sites (Kis = 0.013 and 0.63 μM, respectively). It is effective in vivo, blocking ischemia-induced neurodegeneration in the CA1 region of the hippocampus of gerbils subjected to bilateral carotid artery occlusion. Eliprodil can also have proarrhythmic actions in hearts under normal conditions.Related product price
- Serotonin hydrochloride
₹4492.38-80300 - 7-Hydroxyisoflavone
₹6170.25-9100 - 119431-25-3
₹7470-60100
![ALPHA-(4-CHLOROPHENYL)-4-[(4-FLUOROPHENYL)METHYL]-1-PIPERIDINEETHANOL](https://img.chemicalbook.com/ProductImageEN/2019-8/small/5cb209a9-e5a3-43fd-9135-752a720bab90.jpg){kind=small}