Mosapride citrate
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- ₹0
- Product name: Mosapride citrate
- CAS: 112885-42-4
- MF: C27H33ClFN3O10
- MW: 614.02
- EINECS:601-211-6
- MDL Number:MFCD00874415
- Synonyms:4-AMINO-5-CHLORO-2-ETHOXY-N-[[4-(4-FLUOROBENZYL)-2-MORPHOLINYL]METHYL]BENZAMIDE CITRATE DIHYDRATE;4-Amino-5-chloro-2-ethoxy-N-[[4-[(4-fluorophenyl)methyl]-2-morpholinyl]methyl]-benzamide 2-hydroxy-1,2,3-propanetricarboxylate;Gasmotin;enzamidecitrate ;yl)methyl)-,2-hydroxy-1,2,3-propanetricarboxylate(1:1) ;4-Amino-5-chloro-2-ethoxy-N-[[4-[(4-fluorophenyl)methyl]-2-morpholinyl]methyl]benzamidecitrate;4-amino-5-chloro-2-ethoxy-N-[[4-[(4-fluorophenyl)methyl]morpholin-2-yl]methyl]benzamide;4-azanyl-5-chloro-2-ethoxy-N-[[4-[(4-fluorophenyl)methyl]morpholin-2-yl]methyl]benzamide
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Properties
Melting point :143-145°
storage temp. :Inert atmosphere,2-8°C
solubility :DMSO (Slightly), Ethanol (Slightly, Sonicated)
form :Solid
color :White to Off-White
Stability :Hygroscopic
CAS DataBase Reference :112885-42-4(CAS DataBase Reference)
storage temp. :Inert atmosphere,2-8°C
solubility :DMSO (Slightly), Ethanol (Slightly, Sonicated)
form :Solid
color :White to Off-White
Stability :Hygroscopic
CAS DataBase Reference :112885-42-4(CAS DataBase Reference)
Safety Information
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Description
Mosapride is an agonist of the serotonin (5-HT) receptor subtype 5-HT4 (Ki = 69.9 nM). It is selective for 5-HT4 over 5-HT1, 5-HT2, dopamine D2, and α1- and α2-adrenergic receptors but acts as a partial antagonist at 5-HT3 (Ki = 1,189 nM). It induces relaxation of precontracted rat esophageal thoracic muscularis mucosa preparations and enhances electrically evoked contractions in isolated guinea pig ileum (EC50s = 208.4 and 73.2 nM, respectively). Mosapride (0.5 and 1 mg/kg, i.v.) increases antral and duodenal, but not ileal or colonic, motility in conscious dogs. It also increases gastric emptying in rats when administered at doses ranging from 0.03 to 30 mg/kg.More related product prices
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