Paliperidone
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- ₹5800 - ₹73999.7
- Product name: Paliperidone
- CAS: 144598-75-4
- MF: C23H27FN4O3
- MW: 426.48
- EINECS:620-493-1
- MDL Number:MFCD00871802
- Synonyms:Paliperidone (Invega);3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-Methyl-;Risperidone EP IMpurity C;Paliperidone 9-Hydroxyrisperidone;9-Hydroxyrisperidone solution;Racemic Paliperidone;4h-pyrido(2,1-a)pyrimidin-4-one,6,7,8,9-tetrahydro-3-(2-(4-(6-fluro-1,2-benzis ;oxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-
5 prices
Selected condition：
Brand
- TCI Chemicals (India)
- Sigma-Aldrich(India)
Package
- 10MG
- 50MG
- 200MG
- 1G
- 1ML
- ManufacturerTCI Chemicals (India)
- Product numberP1897
- Product descriptionPaliperidone
- Packaging200MG
- Price₹5800
- Updated2022-05-26
- Buy
- ManufacturerTCI Chemicals (India)
- Product numberP1897
- Product descriptionPaliperidone
- Packaging1G
- Price₹10200
- Updated2022-05-26
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberP0099
- Product descriptionPaliperidone ≥98% (HPLC)
- Packaging10MG
- Price₹18532.4
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberH-076
- Product description9-Hydroxyrisperidone solution 1.0?mg/mL in methanol, ampule of 1?mL, certified reference material, Cerilliant?
- Packaging1ML
- Price₹18659.9
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberP0099
- Product descriptionPaliperidone ≥98% (HPLC)
- Packaging50MG
- Price₹73999.7
- Updated2022-06-14
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| TCI Chemicals (India) | P1897 | Paliperidone | 200MG | ₹5800 | 2022-05-26 | Buy |
| TCI Chemicals (India) | P1897 | Paliperidone | 1G | ₹10200 | 2022-05-26 | Buy |
| Sigma-Aldrich(India) | P0099 | Paliperidone ≥98% (HPLC) | 10MG | ₹18532.4 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | H-076 | 9-Hydroxyrisperidone solution 1.0?mg/mL in methanol, ampule of 1?mL, certified reference material, Cerilliant? | 1ML | ₹18659.9 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | P0099 | Paliperidone ≥98% (HPLC) | 50MG | ₹73999.7 | 2022-06-14 | Buy |
Properties
Melting point :158-160°C
Boiling point :612.3±65.0 °C(Predicted)
Density :1.45±0.1 g/cm3(Predicted)
Flash point :9℃
storage temp. :2-8°C
solubility :DMSO: soluble2mg/mL, clear (warmed)
pka :13.00±0.60(Predicted)
form :powder
color :white to brown
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.
InChI :InChI=1S/C23H27FN4O3/c1-14-17(23(30)28-9-2-3-19(29)22(28)25-14)8-12-27-10-6-15(7-11-27)21-18-5-4-16(24)13-20(18)31-26-21/h4-5,13,15,19,29H,2-3,6-12H2,1H3
InChIKey :PMXMIIMHBWHSKN-UHFFFAOYSA-N
SMILES :C12C(O)CCCN1C(=O)C(CCN1CCC(C3C4=C(ON=3)C=C(F)C=C4)CC1)=C(C)N=2
CAS DataBase Reference :144598-75-4(CAS DataBase Reference)
Boiling point :612.3±65.0 °C(Predicted)
Density :1.45±0.1 g/cm3(Predicted)
Flash point :9℃
storage temp. :2-8°C
solubility :DMSO: soluble2mg/mL, clear (warmed)
pka :13.00±0.60(Predicted)
form :powder
color :white to brown
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.
InChI :InChI=1S/C23H27FN4O3/c1-14-17(23(30)28-9-2-3-19(29)22(28)25-14)8-12-27-10-6-15(7-11-27)21-18-5-4-16(24)13-20(18)31-26-21/h4-5,13,15,19,29H,2-3,6-12H2,1H3
InChIKey :PMXMIIMHBWHSKN-UHFFFAOYSA-N
SMILES :C12C(O)CCCN1C(=O)C(CCN1CCC(C3C4=C(ON=3)C=C(F)C=C4)CC1)=C(C)N=2
CAS DataBase Reference :144598-75-4(CAS DataBase Reference)
Safety Information
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| Signal word: | Danger | ||||||||||||||
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Description
Paliperidone is a potent antagonist of dopamine receptors (IC50s = 1.0 and 0.9 nM for D2 and D3, respectively). It also avidly binds α1- and α2-adrenergic receptors, histamine H1 receptor, and serotonin (5-HT) receptors 5-HT1D and 5-HT2A (Kis = 10, 80, 3.4, 19, 1.2 nM, respectively). Paliperidone is also known as 9-hydroxy risperidone and is the major metabolite of the antipsychotic medication risperidone .Related product price
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