pristimerin
|
- ₹9490 - ₹96916.23
- Product name: pristimerin
- CAS: 1258-84-0
- MF: C30H40O4
- MW: 464.64
- EINECS:251-228-4
- MDL Number:MFCD01711331
- Synonyms:pristimerin;3-Hydroxy-2-oxo-24-nor-D:A-friedoolean-1(10),3,5,7-tetren-29-oic acid methyl ester;Celastrol-methylether;(9β,13α,14β,20α)-3-Hydroxy-9,13-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oicacidmethylester;(9b,13a,14b,20a)-3-Hydroxy-9,13-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tertraen-29-oic acid methyl ester;3-hydroxy-9β,13α-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid, methyl ester;Celastrol methyl ester;Pristimerin(NSC 99281)
3 prices
Selected condition：
Brand
- Sigma-Aldrich(India)
Package
- 5MG
- 25MG
- ManufacturerSigma-Aldrich(India)
- Product number530070
- Product descriptionPristimerin - CAS 1258-84-0 - Calbiochem A cell-permeable plant dienone-phenolic triterpenoid, naturally isolated from tripterygium wilfordii.
- Packaging5MG
- Price₹9490
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberP0020
- Product descriptionPristimerin
- Packaging5MG
- Price₹24183.05
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberP0020
- Product descriptionPristimerin
- Packaging25MG
- Price₹96916.23
- Updated2022-06-14
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Sigma-Aldrich(India) | 530070 | Pristimerin - CAS 1258-84-0 - Calbiochem A cell-permeable plant dienone-phenolic triterpenoid, naturally isolated from tripterygium wilfordii. | 5MG | ₹9490 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | P0020 | Pristimerin | 5MG | ₹24183.05 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | P0020 | Pristimerin | 25MG | ₹96916.23 | 2022-06-14 | Buy |
Properties
Melting point :219.5°C
Boiling point :488.1°C (rough estimate)
Density :1.0271 (rough estimate)
refractive index :1.4800 (estimate)
storage temp. :-20°C
solubility :DMSO: ≥5mg/mL
form :Red solid
pka :8.60±0.70(Predicted)
color :orange
Boiling point :488.1°C (rough estimate)
Density :1.0271 (rough estimate)
refractive index :1.4800 (estimate)
storage temp. :-20°C
solubility :DMSO: ≥5mg/mL
form :Red solid
pka :8.60±0.70(Predicted)
color :orange
Safety Information
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Description
Monoacylglycerol lipase (MAGL) hydrolyzes the endogenous cannabinoid 2-arachidonoyl glycerol (2-AG), terminating its capacity to activate cannabinoid receptors. Pristimerin is a naturally occurring terpenoid that potently inhibits MAGL (IC50 = 93 nM). Its actions are rapid, reversible, and noncompetitive. Pristimerin (1 μM) significantly increases 2-AG levels in isolated rat neurons, indicating that it inhibits endogenous MAGL in cultured cells. Moreover, it does not increase levels of palmitoyl ethanolamide, suggesting that pristimerin does not affect the activity of fatty acid amide hydrolase (FAAH).More related product prices
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