Azelnidipine
- CAS No.
- 123524-52-7
- Chemical Name:
- Azelnidipine
- Synonyms
- CS-905;CS-499;RS-9054;Calblock;Azelpine;Azedipine;Azelidipine;Azenildipine;AZELNIDIPINE;AZELINIDIPINE
- CBNumber:
- CB1781980
- Molecular Formula:
- C33H34N4O6
- Molecular Weight:
- 582.65
- MOL File:
- 123524-52-7.mol
- Modify Date:
- 2024/4/18 11:58:16
| Melting point | 120-126°C |
|---|---|
| Boiling point | 709.3±60.0 °C(Predicted) |
| Density | 1.33±0.1 g/cm3(Predicted) |
| storage temp. | Keep in dark place,Inert atmosphere,Room temperature |
| solubility | DMSO: >10mg/mL |
| pka | 7.89(at 25℃) |
| form | powder |
| color | Yellow |
| Merck | 14,907 |
| InChIKey | ZKFQEACEUNWPMT-UHFFFAOYSA-N |
| CAS DataBase Reference | 123524-52-7(CAS DataBase Reference) |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |   GHS05,GHS07 |
|||||||||
|---|---|---|---|---|---|---|---|---|---|---|
| Signal word | Danger | |||||||||
| Hazard statements | H302-H318 | |||||||||
| Precautionary statements | P280-P301+P312+P330-P305+P351+P338+P310 | |||||||||
| Hazard Codes | Xn | |||||||||
| Risk Statements | 22-41 | |||||||||
| Safety Statements | 26-39 | |||||||||
| WGK Germany | 3 | |||||||||
| RTECS | US7968332 | |||||||||
| HS Code | 2933.79.1500 | |||||||||
| Toxicity | LD50 in female, male mice, female, male rats (mg/kg): 785, 979, 1267, 1971 orally | |||||||||
| NFPA 704 |
|
Azelnidipine price More Price(4)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich(India) | A7106 | Azelnidipine ≥98% (HPLC), powder | 123524-52-7 | 10MG | ₹15631.3 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | A7106 | Azelnidipine ≥98% (HPLC), powder | 123524-52-7 | 50MG | ₹74551.78 | 2022-06-14 | Buy |
| TCI Chemicals (India) | A2433 | Azelnidipine | 123524-52-7 | 1G | ₹7500 | 2022-05-26 | Buy |
| TCI Chemicals (India) | A2433 | Azelnidipine | 123524-52-7 | 5G | ₹14500 | 2022-05-26 | Buy |
Azelnidipine Chemical Properties,Uses,Production
Chemical Properties
Yellow Solid
Uses
Azelnidipine is a dihydropyridine calcium channel blocker with antihypertensice activity. Azelnidipine is used for treating ischemic heart disease and cardiac remodeling after myocardial infarction. S tudies show that Azelnidipine ttreatment can reduce the risk of hyperglycemia induced metabolic disorders
Application
Azelnidipine is a novel dihydropyridine derivative, a L-type calcium channel blocker, and an antihypertensive. Acute administration of azelnidipine prevents a sudden drop of cardiac function after acute stress. Azelnidipine may have a protective role in inflammation associated with atherosclerosis.
Biological Activity
Azelnidipine, a novel dihydropyridine derivative, is a L-type calcium channel blocker and antihypertensive. Unlike other L-type calcium channel blockers, azelnidipine causes minimal stimulation of the sympathetic nervous system despite its significant depressor effect. Azelnidipine may have a protective role in inflammation in atherosclerosis.
Azelnidipine Preparation Products And Raw materials
Raw materials
Preparation Products
Global( 383)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | Inquiry |
|---|---|---|---|---|---|
| Anant Pharmaceuticals Pvt Ltd | +91-8550986868 +91-9485998001 | Haryana, India | 461 | 58 | Inquiry |
| Honour Lab Limited | +919845977466 | Telangana, India | 164 | 58 | Inquiry |
| Hetero Drugs Limited | +91-4023704923 +91-4023704923 | Telangana, India | 296 | 58 | Inquiry |
| Precise Biopharma Pvt Ltd | +91-2267828600 +91-2267828600 | Maharashtra, India | 46 | 58 | Inquiry |
| Afton Pharma | +91-9712000202 +91-9712000202 | Gujarat, India | 63 | 58 | Inquiry |
| Ralington Pharma | +91-7948911722 +91-9687771722 | Gujarat, India | 1350 | 58 | Inquiry |
| Sudarshan Pharma Industries Limited. | 91-22-42221111 | Maharashtra, India | 158 | 58 | Inquiry |
| Indexim International | 08048971004 | Gujarat, India | 112 | 58 | Inquiry |
| Oceanic Pharmachem Pvt. Ltd. | 91-22-42128600 | Maharashtra, India | 2006 | 58 | Inquiry |
| Afton Pharma | 91-9712000202 | Gujarat, India | 40 | 58 | Inquiry |
| Supplier | Advantage |
|---|---|
| Anant Pharmaceuticals Pvt Ltd | 58 |
| Honour Lab Limited | 58 |
| Hetero Drugs Limited | 58 |
| Precise Biopharma Pvt Ltd | 58 |
| Afton Pharma | 58 |
| Ralington Pharma | 58 |
| Sudarshan Pharma Industries Limited. | 58 |
| Indexim International | 58 |
| Oceanic Pharmachem Pvt. Ltd. | 58 |
| Afton Pharma | 58 |
123524-52-7(Azelnidipine)Related Search:
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AZELNIDIPINE
3-[1-(Diphenylmethyl)-3-azetidinyl]-5-(1-methylethyl-2-amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylate
AzelnidipineC33H34N406
AZELINIDIPINE
AZELNIDIPINE(FORR&DONLY)
CS-905, RS-9054, 2-Amino-1,4-dihydro-6-methyl-4-(3 nitrophenyl)-3,5-pyridinedicarboxylic acid 3-[1-(diphenylmethyl)-3-azetidinyl] 5-(1-methylethyl) ester
Azelidipine
Azenildipine
Calblock
CS-905
2-amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic acid 3-[1-(diphenylmethyl)-3-azetidinyl] 5-(methylethyl) ester
(±)-2-AMino-1,4-dihydro-6-Methyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic Acid 3-[1-(DiphenylMethyl)-3-azetidinyl] 5-(1-Methylethyl) Ester
Calblock 3-[1-(DiphenylMethyl)-3-azetidinyl] 5-isopropyl (±)-2-AMino-1,4-dihyd
Azelnidipine (Crystalline forM α)
3-(1-Benzhydrylazetidin-3-yl) 5-isopropyl 2-aMino-6-Methyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate
Azelnidipine, >=99%
3-(1-Benzhydrylazetidin-3-yl) 5-isopropyl 2-amino-6-methyl-4-(3-nitrophenyl)-1,4-dihydropyridine-
Azelnidipine USP/EP
3,5-Pyridinedicarboxylic acid, 2-amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-, 3-[1-(diphenylmethyl)-3-azetidinyl] 5-(1-methylethyl) ester
Azelnidipine 2-Amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic acid 3-[1-(diphenylmethyl)-3-azetidinyl] 5-(methylethyl) ester
RS-9054
3-(1-Benzhydrylazetidin-3-yl) 5-isopropyl 2-amino-6-methyl-4-(3-nitrophenyl)-1,4-dihydropyridi
2-amino-6-methyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylic acid O3-[1-(diphenylmethyl)-3-azetidinyl] ester O5-propan-2-yl ester
CS-499
Azelnidipine Azelnidipine
Azelnidipine >
2-Amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic Acid 3-[1-(Diphenylmethyl)-3-azetidinyl] 5-Isopropyl Ester
3-[1-(Diphenylmethyl)-3-azetidinyl] 5-Isopropyl 2-Amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylate
Azelnidipine USP/EP/BP
Azelnidipine (UR12592, CS-905, CCRIS-8650)
AzelnidipineQ: What is
Azelnidipine Q: What is the CAS Number of
Azelnidipine Q: What is the storage condition of
Azelnidipine Q: What are the applications of
Azelnidipine
Fold the horizon
Azedipine
Azelnidipine Reference Standard
Azelnidipine, ≥ 98.0%
Azelnidipine powder
Azelpine
123524-52-7
23524-52-7
C33H34N4O6
Inhibitors
Cardiovascular Drugs
API