N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide
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- ₹28491.4 - ₹111053.68
- Product name: N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide
- CAS: 942206-85-1
- MF: C28H32Cl2N4O6S2
- MW: 655.61
- EINECS:
- MDL Number:MFCD12912413
- Synonyms:N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide;(N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide;GSK1016790A;GSK101;GSK1016790A;GSK-1016790A;GSK 1016790A;CS-2774;GSK-1016790A;GSK 1016790A;Benzo[b]thiophene-2-carboxamide, N-[(1S)-1-[[4-[(2S)-2-[[(2,4-dichlorophenyl)sulfonyl]amino]-3-hydroxy-1-oxopropyl]-1-piperazinyl]carbonyl]-3-methylbutyl]-
2 prices
Selected condition:
Brand
- Sigma-Aldrich(India)
Package
- 10MG
- 50MG
- ManufacturerSigma-Aldrich(India)
- Product numberG0798
- Product descriptionGSK1016790A ≥98% (HPLC)
- Packaging10MG
- Price₹28491.4
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberG0798
- Product descriptionGSK1016790A ≥98% (HPLC)
- Packaging50MG
- Price₹111053.68
- Updated2022-06-14
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
Sigma-Aldrich(India) | G0798 | GSK1016790A ≥98% (HPLC) | 10MG | ₹28491.4 | 2022-06-14 | Buy |
Sigma-Aldrich(India) | G0798 | GSK1016790A ≥98% (HPLC) | 50MG | ₹111053.68 | 2022-06-14 | Buy |
Properties
Melting point :>119°C (dec.)
Density :1.426±0.06 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: >10mg/mL
form :white solid
pka :8.29±0.50(Predicted)
color :White to Off-White
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.
Density :1.426±0.06 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: >10mg/mL
form :white solid
pka :8.29±0.50(Predicted)
color :White to Off-White
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.
Safety Information
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Description
Transient receptor potential vanilloid 4 (TRPV4) is a nonselective cation channel thought to be involved in osmoregulation, hyperalgesia, and control of epithelial cell volume. GSK1016790A is a TRPV4 agonist that has been reported to elicit calcium influx in HEK cells expressing mouse or human TRPV4 (EC50s = 18 and 2.1 nM, respectively). It has been used to demonstrate a role for TRPV4 in regulating urinary bladder activity and endothelial control of vascular tone.More related product prices
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