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Glucagon Receptor Antagonist I

Glucagon Receptor Antagonist I Structure
  • ₹0
  • Product name: Glucagon Receptor Antagonist I
  • CAS: 438618-32-7
  • MF: C20H30N2OS
  • MW: 346.53
  • EINECS:
  • MDL Number:MFCD01920208
  • Synonyms:Glucagon Receptor Antagonist I;N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide;Butanamide, N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-2-ethyl-;hGCGR Antagonist
Properties Safety Information Description
Manufacturer Product number Product description Packaging Price Updated Buy

Properties

Boiling point :517.8±50.0 °C(Predicted)
Density :1.07±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO: soluble
form :White crystalline solid.
pka :13.46±0.40(Predicted)

Safety Information

Symbol(GHS):
Signal word:
Hazard statements:
Code Hazard statements Hazard class Category Signal word Pictogram P-Codes
Precautionary statements:

Description

Glucagon Receptor Antagonist I is a potent and selective cell-permeable thienyl-amide compound that acts as a competitive antagonist of the glucagon receptor. Exhibits binding to hGCGR with high affinity and prevents its interaction with glucagon (IC50 = 181 nM, KDB = 81 nM, and pA2 = 7.1 in membranes prepared from CHO-hGCGR). Also suppresses glucagon-induced glycogenolysis in human primary hepatocytes and in mice (50 mg/kg, ip).

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Suppliers and manufacturers

Aladdin Scientific Shanghai Aladdin Biochemical Technology Co.,Ltd. EvoBlocks, Ltd. Manchester Organics Shanghai Hao Zhun Biological Technology Co., Ltd. ChemeGen(Shanghai) Biotechnology Co.,Ltd. TargetMol Chemicals Inc. Cayman Chemical Company Shanghai EFE Biological Technology Co., Ltd. Nantong QuanYi Biotechnology Co., Ltd