Entospletinib (GS-9973)
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- Product name: Entospletinib (GS-9973)
- CAS: 1229208-44-9
- MF: C23H21N7O
- MW: 411.46
- EINECS:-0
- MDL Number:MFCD28099806
- Synonyms:GS-9973;6-(1H-Indazol-6-yl)-N-[4-(4-morpholinyl)phenyl]imidazo[1,2-a]pyrazin-8-amine;Entospletinib (GS-9973);Entospletinib Dimesylate;GS-9973, Entospletinib;GS-9973;GS 9973;CS-1602;GS9973; GS 9973; ENTOSPLETINIB
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Properties
Density :1.45±0.1 g/cm3(Predicted)
storage temp. :Desiccate at -20°C
solubility :insoluble in EtOH; insoluble in H2O; ≥20.55 mg/mL in DMSO
form :solid
pka :12.54±0.40(Predicted)
color :White to gray
storage temp. :Desiccate at -20°C
solubility :insoluble in EtOH; insoluble in H2O; ≥20.55 mg/mL in DMSO
form :solid
pka :12.54±0.40(Predicted)
color :White to gray
Safety Information
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Description
Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor with IC50 of 7.7 nM in a cell-free assay and showed 13-to >1000-fold cellular selectivity for Syk over other kinases(including Jak2, ckit, Flt3, Ret, KDR) as assessed by target protein phosphorylation or functional response.More related product prices
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