SB 242084 (hydrochloride)
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- ₹0
- Product name: SB 242084 (hydrochloride)
- CAS: 1049747-87-6
- MF: C21H21Cl3N4O2
- MW: 467.77604
- EINECS:
- MDL Number:
- Synonyms:SB 242084 (hydrochloride);SB-242084 HCl salt;CAS 1049747-87-6;SB242084;SB 242084;CAS 1049747-87-6;SB 242084 2HCL
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
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Properties
storage temp. :Sealed in dry,Room Temperature
solubility :Ethanol:1.0(Max Conc. mg/mL);2.14(Max Conc. mM)
PBS (pH 7.2):10.0(Max Conc. mg/mL);21.38(Max Conc. mM)
DMSO:59.63(Max Conc. mg/mL);127.47(Max Conc. mM)
DMF:30.0(Max Conc. mg/mL);64.13(Max Conc. mM) form :A crystalline solid
color :Off-white to light yellow
solubility :Ethanol:1.0(Max Conc. mg/mL);2.14(Max Conc. mM)
PBS (pH 7.2):10.0(Max Conc. mg/mL);21.38(Max Conc. mM)
DMSO:59.63(Max Conc. mg/mL);127.47(Max Conc. mM)
DMF:30.0(Max Conc. mg/mL);64.13(Max Conc. mM) form :A crystalline solid
color :Off-white to light yellow
Safety Information
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Description
Serotonin (5-hydroxytryptamine, 5-HT) is a neurotransmitter that activates specific receptors located primarily in the gut and central nervous system. SB-242084 is an antagonist of the 5-HT2C receptor (pKi = 9.0), with at least 100-fold more selectivity over other 5-HT, dopamine, or adrenergic receptors. In vivo, it is brain penetrant and has significant anxiolytic activity, without sedative, proconvulsant, or hyperphagic properties. SB-242084 has been used extensively in animal research to evaluate, for example, 5-HT2C receptor agonists and neurotransmitter receptor interactions in mice.Related product price
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Suppliers and manufacturers
A.J Chemicals
InvivoChem
Nantong HI-FUTURE Biology Co., Ltd.
Wuhan Topule Biopharmaceutical Co., Ltd
Aladdin Scientific
Amadis Chemical Company Limited
Shanghai Chaoyan Biotechnology Co., Ltd.
Shanghai Hao Biological Technology Co., Ltd.
Shanghai Jijin Chemical Technology Co., Ltd.
Shenzhen Xinbosheng Biological Technology Co., Ltd.