KENPAULLONE
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- ₹8800 - ₹48755.8
- Product name: KENPAULLONE
- CAS: 142273-20-9
- MF: C16H11BrN2O
- MW: 327.18
- EINECS:
- MDL Number:MFCD02683595
- Synonyms:9-Bromo-7,12-dihydro-indolo[3,2-d][1]benzazepin-6(5H)-one, NSC 664704;9-BroMopaullone;Kenpaullon;9-BROMO-7,12-DIHYDRO-INDOLO[3,2-D][1]BENZAZEPIN-6(5H)-ONE;8-BROMO-7,12-DIHYDRO-INDOLO[3,2-D][1]-BENZAZEPIN-6(5H)-ONE;KENPAULLONE;NSC-664704;Kenpaullone 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one
5 prices
Selected condition：
Brand
- TCI Chemicals (India)
- Sigma-Aldrich(India)
Package
- 1MG
- 5MG
- 10MG
- 50MG
- ManufacturerTCI Chemicals (India)
- Product numberK0052
- Product descriptionKenpaullone
- Packaging10MG
- Price₹8800
- Updated2022-05-26
- Buy
- ManufacturerTCI Chemicals (India)
- Product numberK0052
- Product descriptionKenpaullone
- Packaging50MG
- Price₹19500
- Updated2022-05-26
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberK3888
- Product descriptionKenpaullone ≥98%
- Packaging1MG
- Price₹12221.43
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product number422000
- Product descriptionKenpaullone - CAS 142273-20-9 - Calbiochem A potent, cell-permeable, and reversible inhibitor of glycogen synthase kinase-3β (IC?? = 230 nM), Lck (IC?? = 470 nM), and cyclin-dependent kinases (
- Packaging1MG
- Price₹13100
- Updated2022-06-14
- Buy
- ManufacturerSigma-Aldrich(India)
- Product numberK3888
- Product descriptionKenpaullone ≥98%
- Packaging5MG
- Price₹48755.8
- Updated2022-06-14
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| TCI Chemicals (India) | K0052 | Kenpaullone | 10MG | ₹8800 | 2022-05-26 | Buy |
| TCI Chemicals (India) | K0052 | Kenpaullone | 50MG | ₹19500 | 2022-05-26 | Buy |
| Sigma-Aldrich(India) | K3888 | Kenpaullone ≥98% | 1MG | ₹12221.43 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | 422000 | Kenpaullone - CAS 142273-20-9 - Calbiochem A potent, cell-permeable, and reversible inhibitor of glycogen synthase kinase-3β (IC?? = 230 nM), Lck (IC?? = 470 nM), and cyclin-dependent kinases ( | 1MG | ₹13100 | 2022-06-14 | Buy |
| Sigma-Aldrich(India) | K3888 | Kenpaullone ≥98% | 5MG | ₹48755.8 | 2022-06-14 | Buy |
Properties
Melting point :>300°C (dec.)
Boiling point :613.0±45.0 °C(Predicted)
Density :1.596±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 18 mg/mL, clear, yellow
pka :14.29±0.20(Predicted)
form :Yellow-brown solid
color :yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChIKey :QQUXFYAWXPMDOE-UHFFFAOYSA-N
CAS DataBase Reference :142273-20-9(CAS DataBase Reference)
Boiling point :613.0±45.0 °C(Predicted)
Density :1.596±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 18 mg/mL, clear, yellow
pka :14.29±0.20(Predicted)
form :Yellow-brown solid
color :yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChIKey :QQUXFYAWXPMDOE-UHFFFAOYSA-N
CAS DataBase Reference :142273-20-9(CAS DataBase Reference)
Safety Information
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Description
Kenpaullone is an ATP-competitive inhibitor of several CDKs (cyclin-dependent kinases) as well as GSK-3β (glycogen synthase kinase 3β). It has been shown to inhibit GSK-3 with an IC50 value of 0.23 μM and CDK1/cyclin B, CDK2/cyclin A, CDK5/p25, and lymphocyte kinase with IC50 values of 0.4, 0.68, 0.85, and 0.47 μM, respectively. Due to the compound’s activity, Kenpaullone is useful in the study of cell cycle regulators. Kenpaullone is an inhibitor of cyclin E, ERK 2 and p35.Related product price
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